메뉴 건너뛰기




Volumn 100, Issue 4, 2004, Pages 956-961

Repeated Dosing with Oral Allosteric Modulator of Adenosine A1 Receptor Produces Tolerance in Rats with Neuropathic Pain

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINO 3 (4 CHLOROBENZOYL) 5,6,7,8 TETRAHYDROBENZOTHIOPHENE; ADENOSINE; ADENOSINE A1 RECEPTOR; BENZOTHIOPHENE DERIVATIVE; RADIOLIGAND; T 62; UNCLASSIFIED DRUG;

EID: 1642307808     PISSN: 00033022     EISSN: None     Source Type: Journal    
DOI: 10.1097/00000542-200404000-00028     Document Type: Article
Times cited : (21)

References (32)
  • 1
    • 0023725934 scopus 로고
    • Pharmacological treatment of neuralgic and neuropathic pain
    • McQuay HJ: Pharmacological treatment of neuralgic and neuropathic pain. Cancer Surv 1988; 7:141-59
    • (1988) Cancer Surv , vol.7 , pp. 141-159
    • McQuay, H.J.1
  • 2
    • 0030827378 scopus 로고    scopus 로고
    • A critical review of controlled clinical trials for peripheral neuropathic pain and complex regional pain syndromes
    • Kingery WS: A critical review of controlled clinical trials for peripheral neuropathic pain and complex regional pain syndromes. Pain 1997; 73:123-39
    • (1997) Pain , vol.73 , pp. 123-139
    • Kingery, W.S.1
  • 3
    • 0032540196 scopus 로고    scopus 로고
    • Adenosine receptor activation and nociception
    • Sawynok J: Adenosine receptor activation and nociception. Eur J Pharmacol 1998; 347:1-11
    • (1998) Eur J Pharmacol , vol.347 , pp. 1-11
    • Sawynok, J.1
  • 4
    • 0033050519 scopus 로고    scopus 로고
    • The safety and efficacy of intrathecal adenosine in patients with chronic neuropathic pain
    • Belfrage M, Segerdahl M, Arner S, Sollevi A: The safety and efficacy of intrathecal adenosine in patients with chronic neuropathic pain. Anesth Analg 1999; 89:136-42
    • (1999) Anesth Analg , vol.89 , pp. 136-142
    • Belfrage, M.1    Segerdahl, M.2    Arner, S.3    Sollevi, A.4
  • 5
    • 0022968939 scopus 로고
    • Cardiovascular effects of adenosine infusion in man and their modulation by dipyridamole
    • Biaggioni I, Onrot J, Hollister AS, Robertson D: Cardiovascular effects of adenosine infusion in man and their modulation by dipyridamole. Life Sci 1986; 39:2229-36
    • (1986) Life Sci , vol.39 , pp. 2229-2236
    • Biaggioni, I.1    Onrot, J.2    Hollister, A.S.3    Robertson, D.4
  • 6
    • 0025012275 scopus 로고
    • Effects of intrathecal injection of the adenosine receptor agonists R-phenylisopropyl-adenosine and N-ethylcarboxamide-adenosine on nociception and motor function in the rat
    • Karlsten R, Gordh TJr, Hartvig P, Post C: Effects of intrathecal injection of the adenosine receptor agonists R-phenylisopropyl-adenosine and N-ethylcarboxamide-adenosine on nociception and motor function in the rat. Anesth Analg 1990; 71:60-4
    • (1990) Anesth Analg , vol.71 , pp. 60-64
    • Karlsten, R.1    Gordh Jr., T.2    Hartvig, P.3    Post, C.4
  • 7
    • 0030440984 scopus 로고    scopus 로고
    • Pharmacology of the spinal adenosine receptor which mediates the antiallodynic action of intrathecal adenosine agonists
    • Lee YW, Yaksh TL: Pharmacology of the spinal adenosine receptor which mediates the antiallodynic action of intrathecal adenosine agonists. J Pharmacol Exp Ther 1996; 277:1642-8
    • (1996) J Pharmacol Exp Ther , vol.277 , pp. 1642-1648
    • Lee, Y.W.1    Yaksh, T.L.2
  • 8
    • 0022472286 scopus 로고
    • Angina pectoris-like pain provoked by intravenous adenosine in healthy volunteers
    • Sylven C, Beermann B, Jonzon B, Brandt R: Angina pectoris-like pain provoked by intravenous adenosine in healthy volunteers. BMJ (Clin Res Ed) 1986; 293:227-30
    • (1986) BMJ (Clin Res Ed) , vol.293 , pp. 227-230
    • Sylven, C.1    Beermann, B.2    Jonzon, B.3    Brandt, R.4
  • 9
    • 0026739165 scopus 로고
    • Spinally-mediated antinociception is induced in mice by an adenosine kinase-, but not by an adenosine deaminase-, inhibitor
    • Keil GJ, DeLander GE: Spinally-mediated antinociception is induced in mice by an adenosine kinase-, but not by an adenosine deaminase-, inhibitor. Life Sci 1992; 51:L171-6
    • (1992) Life Sci , vol.51
    • Keil, G.J.1    DeLander, G.E.2
  • 10
    • 0030603728 scopus 로고    scopus 로고
    • Adenosine kinase inhibitors augment release of adenosine from spinal cord slices
    • Golembiowska K, White TD, Sawynok J: Adenosine kinase inhibitors augment release of adenosine from spinal cord slices. Eur J Pharmacol 1996; 307:157-62
    • (1996) Eur J Pharmacol , vol.307 , pp. 157-162
    • Golembiowska, K.1    White, T.D.2    Sawynok, J.3
  • 11
    • 0032995813 scopus 로고    scopus 로고
    • Exogenous and endogenous adenosine enhance the spinal antiallodynic effects of morphine in a rat model of neuropathic pain
    • Lavand'homme PM, Eisenach JC: Exogenous and endogenous adenosine enhance the spinal antiallodynic effects of morphine in a rat model of neuropathic pain. Pain 1999; 80:31-6
    • (1999) Pain , vol.80 , pp. 31-36
    • Lavand'Homme, P.M.1    Eisenach, J.C.2
  • 12
    • 0029816510 scopus 로고    scopus 로고
    • PD 81,723, an allosteric enhancer of the A1 adenosine receptor, lowers the threshold for ischemic preconditioning in dogs
    • Mizumura T, Auchampach JA, Linden J, Bruns RF, Gross GJ: PD 81,723, an allosteric enhancer of the A1 adenosine receptor, lowers the threshold for ischemic preconditioning in dogs. Circ Res 1996; 79:415-23
    • (1996) Circ Res , vol.79 , pp. 415-423
    • Mizumura, T.1    Auchampach, J.A.2    Linden, J.3    Bruns, R.F.4    Gross, G.J.5
  • 13
    • 0035863033 scopus 로고    scopus 로고
    • Differential effects of the allosteric enhancer (2-amino-4,5-dimethyl-trienyl)[3-trifluoromethyl) phenyl-]methanone (PD81,723) on agonist and antagonist binding and function at the human wild-type and a mutant (T277A) adenosine A1 receptor
    • Kourounakis A, Visser C, de Groote M, IJzerman AP: Differential effects of the allosteric enhancer (2-amino-4,5-dimethyl-trienyl)[3-trifluoromethyl) phenyl-]methanone (PD81,723) on agonist and antagonist binding and function at the human wild-type and a mutant (T277A) adenosine A1 receptor. Biochem Pharmacol 2001; 61:137-44
    • (2001) Biochem Pharmacol , vol.61 , pp. 137-144
    • Kourounakis, A.1    Visser, C.2    De Groote, M.3    Ijzerman, A.P.4
  • 14
    • 0025603686 scopus 로고
    • Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes
    • Bruns RF, Fergus JH: Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes. Mol Pharmacol 1990; 38:939-49
    • (1990) Mol Pharmacol , vol.38 , pp. 939-949
    • Bruns, R.F.1    Fergus, J.H.2
  • 15
    • 0034899555 scopus 로고    scopus 로고
    • Allosteric adenosine modulation to reduce allodynia
    • Pan HL, Xu Z, Leung E, Eisenach JC: Allosteric adenosine modulation to reduce allodynia. ANESTHESIOLOGY 2001; 95:416-20
    • (2001) Anesthesiology , vol.95 , pp. 416-420
    • Pan, H.L.1    Xu, Z.2    Leung, E.3    Eisenach, J.C.4
  • 16
    • 0036276780 scopus 로고    scopus 로고
    • Spinal noradrenergic activation mediates allodynia reduction from an allosteric adenosine modulator in a rat model of neuropathic pain
    • Li X, Conklin D, Ma W, Zhu X, Eisenach JC: Spinal noradrenergic activation mediates allodynia reduction from an allosteric adenosine modulator in a rat model of neuropathic pain. Pain 2002; 97:117-25
    • (2002) Pain , vol.97 , pp. 117-125
    • Li, X.1    Conklin, D.2    Ma, W.3    Zhu, X.4    Eisenach, J.C.5
  • 17
    • 0026329329 scopus 로고
    • Sympathectomy alleviates mechanical allodynia in an experimental animal model for neuropathy in the rat
    • Kim SH, Chung JM: Sympathectomy alleviates mechanical allodynia in an experimental animal model for neuropathy in the rat. Neurosci Lett 1991; 134:131-4
    • (1991) Neurosci Lett , vol.134 , pp. 131-134
    • Kim, S.H.1    Chung, J.M.2
  • 19
    • 0017036162 scopus 로고
    • Chronic catheterization of the spinal subarachnoid space
    • Yaksh TL, Rudy TA: Chronic catheterization of the spinal subarachnoid space. Physiol Behav 1976; 7:1032-6
    • (1976) Physiol Behav , vol.7 , pp. 1032-1036
    • Yaksh, T.L.1    Rudy, T.A.2
  • 21
    • 0027980388 scopus 로고
    • Therapeutic time window and dose response of the beneficial effects of ketamine in experimental head injury
    • Shapira Y, Lam AM, Eng CC, Laohaprasit V, Michel M: Therapeutic time window and dose response of the beneficial effects of ketamine in experimental head injury. Stroke 1994; 25:1637-43
    • (1994) Stroke , vol.25 , pp. 1637-1643
    • Shapira, Y.1    Lam, A.M.2    Eng, C.C.3    Laohaprasit, V.4    Michel, M.5
  • 22
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford MM: A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal. Biochem 1976; 72:248-54
    • (1976) Anal Biochem , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 25
    • 0034814354 scopus 로고    scopus 로고
    • Systemic adenosine infusions alleviated neuropathic pain
    • Gyllenhammar E, Nordfors LO: Systemic adenosine infusions alleviated neuropathic pain. Pain 2001; 94:121-2
    • (2001) Pain , vol.94 , pp. 121-122
    • Gyllenhammar, E.1    Nordfors, L.O.2
  • 26
    • 0031738126 scopus 로고    scopus 로고
    • Reduced anti-allodynic effect of the adenosine A1-receptor agonist R-phenylisopropyladenosine on repeated intrathecal administration and lack of cross-tolerance with morphine in a rat model of central pain
    • von Heijne M, Hao JX, Yu W, Sollevi A, Xu XJ, Wiesenfeld-Hallin Z: Reduced anti-allodynic effect of the adenosine A1-receptor agonist R-phenylisopropyladenosine on repeated intrathecal administration and lack of cross-tolerance with morphine in a rat model of central pain. Anesth Analg 1998; 87:1367-71
    • (1998) Anesth Analg , vol.87 , pp. 1367-1371
    • Von Heijne, M.1    Hao, J.X.2    Yu, W.3    Sollevi, A.4    Xu, X.J.5    Wiesenfeld-Hallin, Z.6
  • 27
    • 0022629144 scopus 로고
    • Cross-tolerance studies between caffeine and (-)-N6-(phenylisopropyl)-adenosine (PIA) in mice
    • Ahlijanian MK, Takemori AE: Cross-tolerance studies between caffeine and (-)-N6-(phenylisopropyl)-adenosine (PIA) in mice. Life Sci 1986; 38:577-88
    • (1986) Life Sci , vol.38 , pp. 577-588
    • Ahlijanian, M.K.1    Takemori, A.E.2
  • 28
    • 0021892992 scopus 로고
    • Effects of (-)-N6-(R-phenylisopropyl)-adenosine (PIA) and caffeine on nociception and morphine-induced analgesia, tolerance and dependence in mice
    • Ahlijanian MK, Takemori AE: Effects of (-)-N6-(R-phenylisopropyl)-adenosine (PIA) and caffeine on nociception and morphine-induced analgesia, tolerance and dependence in mice. Eur J Pharmacol 1985; 112:171-9
    • (1985) Eur J Pharmacol , vol.112 , pp. 171-179
    • Ahlijanian, M.K.1    Takemori, A.E.2
  • 29
    • 0028201349 scopus 로고
    • Repeated administration of selective adenosine A1 and A2 receptor agonists in the spontaneously hypertensive rat: Tolerance develops to A1-mediated hemodynamic effects
    • Casati C, Monopoli A, Dionisotti S, Zocchi C, Bonizzoni E, Ongini E: Repeated administration of selective adenosine A1 and A2 receptor agonists in the spontaneously hypertensive rat: Tolerance develops to A1-mediated hemodynamic effects. J Pharmacol Exp Ther 1994; 268:1506-11
    • (1994) J Pharmacol Exp Ther , vol.268 , pp. 1506-1511
    • Casati, C.1    Monopoli, A.2    Dionisotti, S.3    Zocchi, C.4    Bonizzoni, E.5    Ongini, E.6
  • 30
    • 0006169580 scopus 로고
    • Morphine receptors as regulators of adenylate cyclase activity
    • Sharma SK, Nirenberg M, Klee WA: Morphine receptors as regulators of adenylate cyclase activity. Proc Natl Acad Sci U S A 1975; 72:590-4
    • (1975) Proc Natl Acad Sci U S A , vol.72 , pp. 590-594
    • Sharma, S.K.1    Nirenberg, M.2    Klee, W.A.3
  • 31
    • 0035869342 scopus 로고    scopus 로고
    • Chronic exposure to nicotine upregulates the human (alpha)4(beta)2 nicotinic acetylcholine receptor function
    • Buisson B, Bertrand D: Chronic exposure to nicotine upregulates the human (alpha)4(beta)2 nicotinic acetylcholine receptor function. J Neurosci 2001; 21:1819-29
    • (2001) J Neurosci , vol.21 , pp. 1819-1829
    • Buisson, B.1    Bertrand, D.2
  • 32
    • 0029895280 scopus 로고    scopus 로고
    • Effects of long-term treatment with the allosteric enhancer, PD81, 723, on Chinese hamster ovary cells expressing recombinant human A1 adenosine receptors
    • Bhattacharya S, Linden J: Effects of long-term treatment with the allosteric enhancer, PD81, 723, on Chinese hamster ovary cells expressing recombinant human A1 adenosine receptors. Mol Pharmacol 1996; 50:104-11
    • (1996) Mol Pharmacol , vol.50 , pp. 104-111
    • Bhattacharya, S.1    Linden, J.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.