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Volumn 13, Issue 8, 2005, Pages 2837-2846

Novel non-steroidal/non-anilide type androgen antagonists: Discovery of 4-substituted pyrrole-2-carboxamides as a new scaffold for androgen receptor ligands

(4) Wakabayashi, Ken Ichi a Miyachi, Hiroyuki a Hashimoto, Yuichi a Tanatani, Aya a

a UNIVERSITY OF TOKYO (Japan)

Author keywords

Androgen; Antagonist; Pyrrole 2 carboxamides

Indexed keywords

ANDROGEN RECEPTOR; ANTIANDROGEN; FLUTAMIDE; N (4 BENZENESULFONYLAMINO 1 METHYLPYRROLE 2 CARBONYL)PYRROLIDINE; N (4 BENZOYLAMINO 1 METHYLPYRROLE 2 CARBONYL)PYRROLIDINE; N (4 BENZYLAMINO 1 METHYLPYRROLE 2 CARBONYL)PYRROLIDINE; N [1 METHYL 4 (2 NITROPHENYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (2 TOLYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (3 NITROPHENYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (3 TOLYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (4 NITROPHENYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (4 TOLYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [1 METHYL 4 (PHENYLAMINO)PYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (2 CHLOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (2 CYANOPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (2 FLUOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (2 METHOXYPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3 CHLOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3 CYANOPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3 FLUOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3 METHOXYPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3,5 DICHLOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (3,5 DIMETHYLPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (4 CHLOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (4 CYANOPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (4 FLUOROPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; N [4 (4 METHOXYPHENYLAMINO) 1 METHYLPYRROLE 2 CARBONYL]PYRROLIDINE; PYRROLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CANCER INHIBITION; CARCINOMA CELL; DRUG ACTIVITY; DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

EID: 15244342943 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2005.02.019 Document Type: Article

Times cited : (25)

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