2-Substituted-4-aryl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,5] oxazocin-5-one as a structurally new NK1 antagonist

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 5, 2005, Pages 1485-1488

  Seto, Shigeki ^a   Tanioka, Asao ^a   Ikeda, Makoto ^a   Izawa, Shigeru ^a  

^a KYORIN PHARMACEUTICAL CO LTD   (Japan)

Author keywords

NK1 antagonist; Pyrimido 4,5 b 1,5 oxazocin 5 one

Indexed keywords

NEUROKININ 1 RECEPTOR ANTAGONIST; OXAZOCINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BLADDER CAPACITY; CHEMICAL REACTION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; GUINEA PIG; NONHUMAN; REACTION ANALYSIS;

STAPHYLOCOCCUS PHAGE 3A;

EID: 13944271836     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.12.089     Document Type: Article

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