Design and synthesis of an optimized positional scanning library of peptoids: Identification of novel multidrug resistance reversal agents

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 6, 2005, Pages 1923-1929

  Masip, Isabel ^a   Cortés, Nuria ^a   Abad, Maria José ^b   Guardiola, Marisa ^a   Pérez Payá, Enrique ^c   Ferragut, José ^b   Ferrer Montiel, Antonio ^b   Messeguer, Angel ^a  

^a DEPARTMENT OF ENVIRONMENTAL CHEMISTRY   (Spain)

^b MIGUEL HERNÁNDEZ UNIVERSITY   (Spain)

^c CSIC   (Spain)

Author keywords

Chemosensitizers; Combinatorial libraries; Peptoids; Positional scanning

Indexed keywords

AMINE; AMINO ACID DERIVATIVE; DAUNORUBICIN; GLYCINE; GLYCOPROTEIN P; MEMBRANE PROTEIN; MONOMER; PEPTOID; UNCLASSIFIED DRUG; VERAPAMIL; [N [2 (2' FLUOROPHENYL)ETHYL]GLYCYL] N [2 (2',4' DICHLOROPHENYL)ETHYL] GLYCINAMIDE; [N [2 (4' FLUOROPHENYL)ETHYL]GLYCYL] N [2 (2',4' DICHLOROPHENYL)ETHYL] GLYCINAMIDE;

AMINATION; AMINO TERMINAL SEQUENCE; ANIMAL CELL; ARTICLE; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SYNTHESIS; GENE FUNCTION; GENE LIBRARY; GENETIC SCREENING; GENETIC VARIABILITY; MOUSE; MULTIDRUG RESISTANCE; NONHUMAN; OBSERVATION; PHARMACOPHORE; PROTEIN STRUCTURE; SOLID;

EID: 13844322495     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.01.024     Document Type: Article

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