Effect of combined histamine H1 and H3 receptor blockade on cutaneous microvascular permeability elicited by compound 48/80

Life Sciences

Volumn 76, Issue 16, 2005, Pages 1787-1794

  McLeod, Robbie L ^a   Mingo, Garfield G ^a   Kreutner, William ^a   Hey, John A ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Antihistamine; Compound 48 80; Evans blue; Histamine H1 antagonist; Histamine H3 antagonist; Urticaria; Wheal and flare

Indexed keywords

CHLORPHENIRAMINE; CLOBENPROPIT; COMPOUND 48-80; HISTAMINE; HISTAMINE H1 RECEPTOR ANTAGONIST; HISTAMINE H3 RECEPTOR ANTAGONIST; THIOPERAMIDE;

ANESTHESIA; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG EFFECT; EXTRAVASATION; GUINEA PIG; HISTAMINE RELEASE; INHIBITION KINETICS; MALE; MICROVASCULATURE; NONHUMAN; SKIN PERMEABILITY; URTICARIA;

ANIMALIA; CAVIA PORCELLUS; SUS SCROFA;

EID: 13444301282     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.lfs.2004.08.033     Document Type: Article

References (37)

1. 3) of histamine receptor Nature 302 1983 832 837
2. S.S. Bleehen, S.E. Thomas, and M.W. Greaves Cimetidine and chlorpheniramine in the treatment of chronic idiopathic urticaria: a multi-centre randomized double-blind study British Journal of Dermatology 117 1987 81 88
3. 3 modulation of nasal airway blood flow and resistance in the cat American Journal of Respiratory and Critical Care 149 1994 A909
4. 3H]-acetylcholine release from slices of rat entorhinal cortex British Journal of Pharmacology 105 1992 919 923
5. C.A. Commens, and M.W. Greaves Cimetidine in chronic idiopathic urticaria: a randomized double-blind study British Journal of Dermatology 99 1978 675 679
6. L.J. Cook, and S.H. Shuster Lack of effect of cimetidine in chronic idiopathetic urticaria Acta Dermato-Venereologica (Stockh) 63 1993 265 267
7. A. Goldberg, M. Shapiro, I. Hammel, and Y.A. Merkori Cutaneous responses to histamine, compound 48/80 and codeine in patients with hyperthyroidism Annals of Allergy 64 1990 179 181
8. 3 receptors British Journal of Pharmacology 107 1992 347 350
9. 3 receptors in the heart Journal of Pharmacology and Experimental Therapeutics 77 1995 206 210
10. S. Kaur, M. Greaves, and N. Eftekhari Fractitious urticaria (dermographia): treatment by cimetidine and chlorpheniramine in a randomized study British Journal of Dermatology 104 1981 185 190
11. 3 receptor agonist R-α- methylhistamine in human skin British Journal of Dermatology 138 1998 622 626
12. D. Lagunoff, T.W. Martin, and G. Read Agents that release histamine from mast cells Annual Review of Pharmacology and Toxicology 23 1983 331 351
13. E. Laurikainen, J.M. Miller, A.L. Nuttall, and W.S. Quirk The vascular mechanism of action of betahistine in the inner ear of the guinea pig European Archives of Oto-rhino-laryngology 255 1998 119 123
14. 3 activation depresses cardiac function in experimental sepsis Journal of Applied Physiology 85 1998 1693 1701
15. 3 receptors-general characterization and their function in the cardiovascular system Journal of Physiology and Pharmacology 49 1998 191 211
16. 3 receptors-mediated inhibition of neurogenic vasopressor responses in the pithed rats European Journal of Pharmacology 205 1991 307 310
17. 2 antagonists Annals of Allergy 50 1983 241 245
18. 2-receptor blocking agent British Journal of Clinical Pharmacology 4 1977 364 369
19. 3 mediated decrease in basal vascular resistance in guinea pigs British Journal of Pharmacology 110 1993 553 558
20. 3 receptors by R-α-methylhistamine in the guinea pig General Pharmacology 27 1996 1001 1007
21. 3 receptor blockade produces nasal decongestion in the cat American Journal of Rhinology 13 1999 391 399
22. 3 antagonists T.T. Hansel P.J. Barnes New Drugs for Asthma, Allergy and COPD vol. 31 2001 Karger Basel 133 136
23. J. Miller, and H.S. Nelson Suppression of immediate skin tests by ranitidine Journal of Allergy and Clinical Immunology 84 1989 895 899
24. 2 antihistamine therapy in chronic urticaria Archives of Dermatology 117 1981 404 407
25. 1 antihistamine therapy in chronic urticaria Annals of Allergy 71 1993 585 591
26. A.D. Ormerod Urticaria, recognition, causes and treatment Drug 48 1994 717 730
27. E. Paul, and R.H. Bodeker Treatment of chronic urticaria with terfenadine and ranitidine. A randomized double-blind study in 45 patients European Journal of Clinical Pharmacology 31 1986 277 280
28. 2 blockers Clinical Allergy 8 1978 429 433
29. J. Ring, K. Brockow, M. Ollert, and R. Engst Antihistamines in urticaria Clinical and Experimental Allergy 29 1999 31 37
30. 3 receptors in isolated guinea pig pulmonary artery and ileum European Journal of Pharmacology 294 1995 329 335
31. 3 receptor-mediated inhibition of serotonin release in the rat brain cortex Naunyn-Schmiedeberg's Archives of Pharmacology 337 1988 588 590
32. 3 receptors Naunyn-Schmiedeberg's Archives of Pharmacology 340 1989 633 638
33. 1-receptor antagonist drugs New England Journal of Medicine 330 1994 1663 1670
34. 1-blockade effect of fexofenadine Annals of Allergy, Asthma and Immunology 79 1997 530 532
35. C.H. Smith, B. Atkinson, R.W. Morris, N. Haynes, J.C. Foreman, and T.H. Lee Cutaneous responses to vasoactive intestinal polypeptide in chronic idiopathic urticaria Lancet 339 1992 91 93
36. S. Tozzi, F.E. Roth, and A. Tabachnick The pharmacology of azatadine, a potential antiallergy drug Agents and Action 4 1974 264 270
37. 3 receptors in human saphenous vein and guinea pig ileum European Journal of Pharmacology 366 1999 73 78