Desensitization Masks Nanomolar Potency of ATP for the P2X1 Receptor

Journal of Biological Chemistry

Volumn 279, Issue 8, 2004, Pages 6426-6433

  Rettinger, Jürgen ^a   Schmalzing, Günther ^b  

^a MAX PLANCK INSTITUTE OF BIOPHYSICS   (Germany)

^b RWTH AACHEN UNIVERSITY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINETRIPHOSPHATE; CHEMICAL ACTIVATION; PHOSPHORUS; REACTION KINETICS;

DESENSITIZATION; NANOMOLAR POTENCY;

BIOCHEMISTRY;

ADENOSINE TRIPHOSPHATE; PURINE P2X1 RECEPTOR; SURAMIN;

ARTICLE; CALCIUM CURRENT; CATION TRANSPORT; CHANNEL GATING; CHIMERA; CROSS LINKING; DESENSITIZATION; HYDROPHOBICITY; NERVE EXCITABILITY; NONHUMAN; POLYACRYLAMIDE GEL ELECTROPHORESIS; PRIORITY JOURNAL; PROTEIN ANALYSIS; RECEPTOR DOWN REGULATION;

ADENOSINE TRIPHOSPHATE; AFFINITY LABELS; ANIMALS; BINDING, COMPETITIVE; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGY; KINETICS; MODELS, BIOLOGICAL; MODELS, CHEMICAL; OOCYTES; PLASMIDS; PROTEIN BINDING; RECEPTORS, PURINERGIC P2; RECOMBINANT FUSION PROTEINS; SURAMIN; THIONUCLEOTIDES; TIME FACTORS; XENOPUS;

EID: 1342282988     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M306987200     Document Type: Article

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