Pyrrolidinohydroquinazolines - A novel class of CCR3 modulators

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 3, 2005, Pages 669-673

  Anderskewitz, Ralf ^a   Bauer, Rolf ^a   Bodenbach, Gisela ^a   Gester, Dirk ^a   Gramlich, Bernd ^a   Morschhäuser, Gerd ^a   Birke, Franz W ^a  

^a BOEHRINGER INGELHEIM PHARMA GMBH AND CO KG   (Germany)

Author keywords

Agonist; Antagonist; CCR3; Eotaxin

Indexed keywords

CHEMOKINE RECEPTOR CCR3; PYRROLIDINOHYDROQUINAZOLINE DERIVATIVE; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG SYNTHESIS; REACTION OPTIMIZATION;

CALCIUM SIGNALING; CHEMOKINES, CC; EOSINOPHILS; HUMANS; QUINAZOLINES; RECEPTORS, CHEMOKINE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 12444330289     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.039     Document Type: Article

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