HIV-1 resistance profile of the novel nucleoside reverse transcriptase inhibitor β-D-2′,3′-dideoxy-2′,3′didehydro-5- fluorocytidine (Reverset™)

Antiviral Chemistry and Chemotherapy

Volumn 14, Issue 1, 2003, Pages 49-59

  Geleziunas, Romas ^b   Gallagher, Karen ^c   Zhang, Hangchun ^b   Bacheler, Lee ^d   Garber, Sena ^e   Wu, Jing Tao ^f   Shi, Guoen ^g   Otto, Michael J ^h   Schinazi, Raymond F ^a   Erickson Viitanen, Susan ^h  

^a EMORY UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

^c Drug Metabolism Pharmacokinetics Clinical Pharmacology   (United States)

^d Tibotec Virco USA   (United States)

^e ASTRAZENECA   (United Kingdom)

^f MILLENNIUM PHARMACEUTICALS INC   (United States)

^g Palatin Technologies   (United States)

^h PHARMASSET INC   (United States)

Author keywords

Multidrug resistance; Nucleoside analogue; Resistance

Indexed keywords

BETA DEXTRO 2',3' DIDEOXY 2',3' DIDEHYDRO 5 FLUOROCYTIDINE; CYTIDINE DERIVATIVE; DIDANOSINE; ELVUCITABINE; LAMIVUDINE; RNA DIRECTED DNA POLYMERASE; RNA DIRECTED DNA POLYMERASE INHIBITOR; TENOFOVIR; UNCLASSIFIED DRUG; ZIDOVUDINE;

ANTIVIRAL ACTIVITY; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYTOPATHOGENIC EFFECT; DRUG EFFICACY; DRUG POTENCY; GENOTYPE; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; IC 50; IN VITRO STUDY; NONHUMAN; PRIORITY JOURNAL; TREATMENT INDICATION; VIRUS ISOLATION; VIRUS MUTANT; VIRUS MUTATION; VIRUS RECOMBINANT; VIRUS REPLICATION; VIRUS RESISTANCE; VIRUS STRAIN;

EID: 12444325183     PISSN: 09563202     EISSN: None     Source Type: Journal    
DOI: 10.1177/095632020301400105     Document Type: Article

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