Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 3, 2005, Pages 567-571

  Innocenti, Alessio ^a   Vullo, Daniela ^a   Scozzafava, Andrea ^a   Supuran, Claudiu T ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BICARBONATE; BISMUTH; BROMATE; CARBONATE DEHYDRATASE INHIBITOR; CARBONIC ACID; CHLORATE; IODATE; ISOENZYME; MEMBRANE PROTEIN; METASILICATE; MITOCHONDRIAL PROTEIN; MOLYBDIC ACID; NITRATE; PERCHLORATE; PERIODATE; SILICATE; SULFAMIC ACID; SULFAMIDATE; SULFATE; UNCLASSIFIED DRUG; VANADIC ACID; ZINC ION;

ACIDITY; ADAPTATION; ARTICLE; BINDING AFFINITY; CHEMICAL BINDING; COMPARATIVE STUDY; ENZYME ACTIVE SITE; ENZYME INHIBITION; EVOLUTION; GEOMETRY; HUMAN; MITOCHONDRION; PH MEASUREMENT; STRUCTURE ANALYSIS;

ANIONS; ANTIGENS, NEOPLASM; CARBON DIOXIDE; CARBONATES; CARBONIC ANHYDRASE I; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASE IV; CARBONIC ANHYDRASE V; CARBONIC ANHYDRASES; HUMANS; HYDROGEN-ION CONCENTRATION; ISOENZYMES; NITRATES; STRUCTURE-ACTIVITY RELATIONSHIP; SULFATES;

EID: 12444317530     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.056     Document Type: Article

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