Celecoxib incorporated chitosan microspheres: In vitro and in vivo evaluation

Journal of Drug Targeting

Volumn 12, Issue 9-10, 2004, Pages 549-557

  Thakkar, Hetal ^a   Sharma, R K ^b   Mishra, A K ^b   Chuttani, Krishna ^b   Murthy, R S R ^a  

^a M S UNIVERSITY OF BARODA   (India)

^b INSTITUTE OF NUCLEAR MEDICINE AND ALLIED SCIENCES   (India)

Author keywords

Biodegradable polymers; Celecoxib; Chitosan; Glutathione

Indexed keywords

CELECOXIB; CHITOSAN; GLUTATHIONE; MICROSPHERE; TECHNETIUM 99M;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG RELEASE; DRUG RETENTION; GAMMA SCINTIGRAPHY; IN VITRO STUDY; IN VIVO STUDY; KNEE ARTHRITIS; MALE; NONHUMAN; PARTICLE SIZE; PRIORITY JOURNAL; RAT;

ANIMALS; CHITOSAN; DRUG EVALUATION, PRECLINICAL; MALE; MICROSPHERES; PARTICLE SIZE; PYRAZOLES; RATS; RATS, SPRAGUE-DAWLEY; SULFONAMIDES;

EID: 11944258052     PISSN: 1061186X     EISSN: None     Source Type: Journal    
DOI: 10.1080/10611860400010630     Document Type: Article

References (39)

1. Akbuga, J. and Bergisadi, N. (1996) "5-Fluorouracil-loaded chitosan microspheres: preparation and release characteristics", J. Microencapsul. 13, 161-168.
2. Akbuga, J. and Bergisadi, N. (1999) "Effect of formulation variables on cis-platin loaded chitosan microsphere properties", J. Microencapsul. 16, 697-703.
3. Ashcroff, D., Chapman, S., Clark, W. and Millson, S. (2001) "Upper gastroduodenal ulceration in arthritis patients treated with celecoxib", Ann. Pharmacother. 35, 829-834.
4. Benacereff, B., Biozzi, G., Halpern, B.N. and Stiffel, C. (1975) In: Halpern, B.N. and Delafresnage, J.F., eds, Physiology of the Reticulo-Endothelial System (PubBlackwell Scientific, Oxford).
5. Banerjee, T., Mitra, S., Singh, A., Sharma, R.K. and Maitra, A. (2002) "Preparation, characterization and biodistribution of ultrafine chitosan nanoparticles", Int. J. Pharm. 243, 93-105.
6. Benita, S., Benoit, J.P., Puisieux, F. and Thies, C. (1984) "Characterization of drug loaded poly (D,L-Lactide) microspheres", J. Pharm. Sci. 73, 1721-1724.
7. Bing, R.J. (2003) "Cyclooxygenase-2 inhibitors: is there an association with coronary or renal events?", Curr. Atherosclerl. Rep. 5, 114-117.
8. Bird, H.A., Ring, E.F., Daniel, R. and Bacon, P.A. (1977) "Comparison of intra-articular methotrexate with intra-articular triamcinolone hexacetonide by thermography", Curr. Med. Res. Opin. 5, 141-146.
9. Bozdag, S., Calis, S., Kas, H.S., Ercan, M.T., Peksoy, L. and Hincal, A. (2001) "In vitro evaluation and intra-articular administration of biodegradable microspheres containing naproxen sodium", J. Microencapsul. 18, 443-456.
10. Brown, K.E., Leong, K., Huang, C.H., Dalal, R., Green, G.D., Haimes, H.B., Jimenez, P.A. and Bathon, J. (1998) "Gelatin /Chondroitin 6 sulphate microspheres for the delivery of therapeutic proteins to the joint", Arthritis Rheum. 41, 2185-2195.
11. Camilleri, J.P., Williams, A.S., Amos, N. and Williams, B.D. (1993) "Uptake of Liposome clodronate compared to free clodronate in inflamed rat paws", Arthritis Rheum. 36(Suppl. 9), S213.
12. Haslett, C., Chilvers, E.R., Hunter, A.A. and Boon, N.A., eds (1999) "Diseases of the connective tissues, joints and bones", Ch. 12, Davidson's Principles and Practice of Medicine (Churchill Livingstone, London), pp 842-845.
13. Denkbas, E.B., Seyyal, M. and Piskin, E. (1999) "5-Fluorouracil loaded chitosan microspheres for chemoembolization", J. Microencapsul. 16, 741-749.
14. Dingle, J.T., Gordon, J.L., Hazleman, B.L., Knight, C.G., Thomas, D.P. and Philips, N.C. (1978) "Novel treatment for joint inflammation", Nature 271, 373.
15. m-glutathione for imaging inflammatory lesions", Nucl. Med. Commun. 15, 533-539.
16. 3H] methotrexate injected into normal or arthritic joints", J. Pharm. Pharmacol. 40, 464-468.
17. Foong, W.C. and Green, K.L. (1993) "Treatment of antigen-induced arthritis in rabbits with liposome entrapped methotrexate injected intra-articularly", J. Pharm. Pharmacol. 45, 204-209.
18. Genta, I., Conti, B., Perugini, P., Pavanetto, F., Spadaro, A. and Puglisi, G. (1997) "Bioadhesive microspheres for ophthalmic administration of acyclovir", J. Pharm. Pharmacol. 49, 737-742.
19. Glutaral disinfectant solution in United states Pharmacopoeia XXII, National Formulary XVII, 1990, pp1934.
20. Horisawa, E., Horita, T., Kawazoe, S., Yamada, J., Yamamoto, H., Takeuchi, H. and Kawashima, Y. (2002) "Prolonged anti-inflammatory action of D,L-lactide/glycolide copolymer nanospheres containing betamethasone sodium phosphate for an intra-articular delivery system in antigen-induced arthritic rabbit", Pharm. Res. 19, 403-410.
21. Jameela, S.R. and Jayakrishnan, A. (1995) "Glutaraldehyde cross-linked chitosan microspheres as a long acting biodegradable drug delivery vehicle: studies on the in vitro release of mitoxantrone and in vivo degradation of microspheres in rat muscle", Biomaterials 16, 769-775.
22. Jameela, S.R., Kumary, T.V., Lal, A.V. and Jayakrishnan, A. (1998) "Progesterone loaded chitosan microspheres: a long acting biodegradable controlled delivery system", J. Control. Release 52, 17-24.
23. Kassab, A.Ch., Xu, K., Denkbas, E.B., Dou, Y., Zhao, S. and Piskin, E. (1997) "Rifampicin carrying polyhydroxybutyrate microspheres as potential chemoembolization agent", J. Biomater. sci. 8, 947-961, Polymer Edition.
24. Kumbhar, S.G., Kulkarni, A.R. and Aminabhavi, T.M. (2002) "Cross-linked chitosan microspheres for encapsulation of diclofenac sodium; effect of cross-linking agent", J. Microencapsul. 19 173-180.
25. Lim, L.Y., Lucy, S.C. and Wan, Thai P.Y. (1997) "Chitosan microspheres prepared by emulsification and ionotropic gelation", Drug Dev. Ind. Pharm. 23, 981-985.
26. Monkkonen, J., Liukkonen, J., Taskinen, M., Heath, T.D. and Urtii, A. (1995) "Studies on liposomal formulations for intra-articular delivery of clodronate", J. Control. release 35, 145-154.
27. Nishioka, Y., Kyotani, S., Okamura, M., Miyazaki, M., Okazaki, K., Ohnishi, S., Yamamoto, Y. and Ito, K. (1990) "Release characteristics of cisplatin chitosan microspheres and effect of containing chitin", Chem. Pharm. Bull. 38, 2871-2873.
28. Noble, J., Jones, A.G., Davies, M.A., Sledge, C.B., Kramer, R.I. and Livni, E. (1983) "Leakage of radioactive particle systems from synovial joint studied with a gamma camera", J. Bone Joint Surg. Am. 65, 381-389.
29. Ratcliffe, J.H., Hunneyball, I.M., Smith, A., Wilson, C.G. and Davis, S.S. (1984) "Preparation and evaluation of biodegradable polymeric systems for the intra-articular delivery of drugs", J. Pharm. Pharmacol. 36, 431-436.
30. Ratcliffe, J.H., Hunneyball, I.M., Smith, A., Wilson, C.G. and Davis, S.S. (1987) "Albumin microspheres for intra-articular drug delivery: investigation of their retention in normal and arthritic knee joints in rabbits", J. Pharm. pharmacol. 28, 290-295.
31. Sansdrap, P. and Moes, A.J. (1993) "Influence of manufacturing parameters on the size characteristics and release profiles on Nifedipine from poly (D, L-lactide-co-glycolide) microspheres", Int. J. pharm. 98, 157-164.
32. Shu, X.Z. and Zhu, K.J. (2001) "Chitosan/gelatin microspheres prepared by modified emulsification and ionotropic gelation", J. Microencapsul. 18, 237-245.
33. Thanoo, B.C., Sunny, M.C. and Jayakrishnan, A. (1992) "Cross-linked chitosan microspheres: preparation and evaluation as a matrix for the controlled release of pharmaceuticals", J. pharm. pharmacol. 44, 283-286.
34. Tuncay, M., Calis, S., Kas, H.S., Ercan, M.T., Peksoy, L. and Hincal, A. (2000a) "In vitro and in vivo evaluation of diclofenac sodium loaded albumin microspheres", J. Microencapsul. 17, 145-155.
35. Tuncay, M., Calis, S., Kas, H.S., Ercan, M.T., Peksoy, L. and Hincal, A. (2000b) "Diclofenac sodium incorporated PLGA (50:50) microspheres:formulation considerations and in vitrolin vivo evaluation", Int. J. Pharm. 195, 179-188.
36. Vogel, G.H. and Vogel, W.H. (eds) (1997) "Methods for testing immunological factors", Drug Discovery and Evaluation-Pharmacological Assays (Springer Verlag, Berlin Heidelberg), p 445.
37. Wallis, W.J., Simkin, P.A. and Nelp, W.B. (1987) "Protein traffic in human synovial effusions", Arthritis Rheum. 30, 57-63.
38. Wang, Y.M., Sato, H., Adachi, I. and Horikoshi, I. (1996) "Optimization of the formulation design of chitosan microspheres containing cisplatin", J. Pharm. Sci. 85, 1204-1210.
39. Woolf, E., Fu, I. and Matuszewski, B. (2000) "Determination of celecoxib in human plasma by normal phase high performance liquid chromatography with column switching and ultraviolet absorbance detection", J. Chromatogr. B Biomed. Sci. Appl. 738, 377-385.