Optimization of pH-independent release of nicardipine hydrochloride extended-release matrix tablets using response surface methodology

International Journal of Pharmaceutics

Volumn 289, Issue 1-2, 2005, Pages 87-95

  Huang, Yaw Bin ^a   Tsai, Yi Hung ^a   Lee, Shu Hui ^a   Chang, Jui Sheng ^a   Wu, Pao Chu ^a  

^a KAOHSIUNG MEDICAL UNIVERSITY   (Taiwan)

Author keywords

Dissolution; Extended release dosage form; Mixture experimental design; Nicardipine response surface methodology

Indexed keywords

ALGINIC ACID; DRUG ADDITIVE; HYDROXYPROPYLMETHYLCELLULOSE; MICROCRYSTALLINE CELLULOSE; NICARDIPINE; POLYMER;

ARTICLE; CHEMICAL COMPOSITION; DRUG DESIGN; DRUG EFFECT; DRUG FORMULATION; DRUG RELEASE; EXPERIMENT; HYDROPHILICITY; KINETICS; MATRIX TABLET; METHODOLOGY; MODEL; PH; PREDICTION; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; RESPONSE SURFACE METHOD; SUSTAINED DRUG RELEASE; TIMED DRUG RELEASE;

ALGINATES; CELLULOSE; CHEMISTRY, PHARMACEUTICAL; GASTRIC JUICE; GLUCURONIC ACID; HEXURONIC ACIDS; HYDROGEN-ION CONCENTRATION; METHYLCELLULOSE; NICARDIPINE; SOLUBILITY; TABLETS, ENTERIC-COATED; TECHNOLOGY, PHARMACEUTICAL; TIME FACTORS;

EID: 11844284788     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2004.10.021     Document Type: Article

References (30)

1. D.R. Abernethy, and J.B. Schwartz Pharmacokinetics of calcium antagonist under development Clin. Pharmacokinet. 15 1988 1 14
2. S. Bouckaert, D.L. Massart, B. Massart, and J.P. Rremon Optimization of a granulation procedure for a hydrophilic matrix tablet design Drug Dev. Ind. Pharm. 22 1996 321 327
3. W.A. Cressman, and D. Summer The dog as a quantitative model for evaluation of nondisintegrating sustained-release tablets J. Pharm. Sci. 60 1971 132 134
4. N.D. Eddington, M. Ashraf, L.L. Augsburger, J.L. Leslie, M.J. Fossler, L.J. Lesko, V.P. Shah, and G.S. Rekhi Identification of formulation and manufacturing variables that influence in vitro dissolution and in vivo bioavialability of nicardipine hydrochloride tablets Pharm. Dev. Technol. 3 1998 535 547
5. L.C. Feely, and S.S. Davis Influence of surfactants on the drug release from hydroxypropylmethylcellulose Int. J. Pharm. 41 1988 83 90
6. C.M. Fernandes, T.M. Vieira, and F.J.B. Veiga Physicochemical characterization and in vitro dissolution behavior of nicardipine-cyclodextrins inclusion compounds Eur. Pharm. Sci. 15 2002 79 88
7. J.L. Ford, M.H. Rubinstein, and J.E. Hogan Formation of sustained release promethazine hydrochloride tablets using hydroxypropylmethylcellulose matrix Int. J. Pharm. 24 1985 327 338
8. P. Gao, and R.H. Meury Swelling of hydroxypropylmethylcellulose matrix tablet Part 1. Characterization of swelling using a novel optical imaging method J. Pharm. Sci. 85 1996 725 731
9. M.C. Gohel, and A.F. Amin Formulation optimization of controlled release diclofenac sodium microspheres using factorial design J. Controlled Release 51 1998 115 122
10. D.J.M. Graham, R.J. Dow, D.J. Hall, D.F. Alexander, and E.J. Mroszczak The metabolism and pharmacokinetics of nicardipine hydrochloride in man Br. J. Clin. Pharmacol. 20 1985 23s 28s
11. A. Hassegawa, R. Kawamura, H. Nakagawa, and I. Sugimata Application of solid dispersion with enteric coating agents to overcome some pharmaceutical problems Chem. Pharm. Bull. 34 1986 2183 2190
12. S. Higuchi, H. Sasaki, and T. Seki Pharmacokinetic studies on nicardipine hydrochloride, a new vasodilator, after repeated administration to rats, dogs and humans Xenobiotica 10 1980 897 903
13. H.O. Ho, L.C. Chen, H.M. Lin, and M.T. Sheu Penetration enhancement by menthol combined with a solubilization effect in a mixed solvent system J. Controlled Release 51 1998 301 311
14. Y.B. Huang, Y.H. Tsai, W.C. Yang, J.S. Chang, P.C. Wu, and K. Takayama Once-daily propranolol extended-release tablet dosage form: formulation design and in vitro/in vivo investigation Eur. J. Pharm. Biopharm. 58 2004 607 614
15. Y.B. Huang, Y.H. Tsai, W.C. Yang, J.S. Chang, and P.C. Wu Optimization of sustained-release propranolol dosage form using factorial design and response surface methodology Biol. Pharm. Bull 27 2004 1626 1629
16. Huang, Y.B., Tsai, Y.H., Sung, C.H., Chang, J.S., Tsai, M.J., Wu, P.C., submitted for publication. Preparation of nicardipine sustained-release dosage form. Arch. Pharm. Res., submitted for publication.
17. A.A. Karnachi, and M.A. Khan Box-Behnken design for the optimization of formulation variables of indomethacin coprecipitates with polymer mixtures Int. J. Pharm. 131 1996 9 17
18. N. Katori, K. Okudaria, N. Aoyagi, Y. Takeda, and M. Uchiyama In vitro and in vivo correlation for controlled-release formulation of d-chlorpheniramine maleate J. Pharmacobio. Dyn. 14 1991 567 575
19. A. Nokhodchi, S. Norouzi-Sani, M.R. Siahi-Shadbad, F. Lotfipoor, and M. Saeedi The effect of various surfactants on the release rate of nicardipine hydrochloride from hydroxypropylmethylcellulose (HPMC)-Eudragit matrix Eur. J. Pharm. Sci. 54 2002 349 356
20. E. Lahdenpaa, M. Niskanen, and J. Yliruusi Crushing strength disintegration time and weight variation of tablets compressed from three AVICEL pH grades and their mixtures Eur. J. Pharm. Biopharm. 42 1997 315 322
21. J.Z. Li, G.S. Rekhi, L.L. Augsburger, and R.F. Shangraw The role of intra- and extragranular microcrystalline cellulose in tablet dissolution Pharm. Dev. Technol. 1 1996 343 355
22. P.L. Ritger, and N.S. Peppas A simple equation for disposition of solute release II: Fickian and anomalous release from swellable devices J. Controlled Release 5 1987 37 42
23. K. Sako, T. Sawada, H. Nakashima, S. Yokohama, and T. Sonobe Influence of water soluble fillers on hydroxypropylmethylcellulose matrix on in vitro and in vivo drug release J. Controlled Release 81 2002 165 172
24. E.M. Sorkin, and S.P. Clissold Nicardipine. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy, in the treatment of angina pectoris, hypertension and related cardiovascular disorders Drugs 33 1987 296 345
25. S.K. Singh, J. Dodge, M.J. Durrani, and M. Khan Factorial design in the feasibility of producing Microcel MC 101 pellets by extrusion spheronization Int. J. Pharm. 115 1995 53 60
26. K. Takayama, and T. Nagai Novel computer optimization methodology for pharmaceutical formulations investigated by using sustained-release granules of indomethacin Chem. Pharm. Bull. 37 1989 160 167
27. T. Uchida, M. Kawata, and S. Goto In vivo evaluation of ethyl cellulose microcapsules containing amipicillin using rabbits, dogs and humans J. Pharmacobio. Dyn. 9 1986 631 637
28. M. Vlachou, N. Hani, M. Efentakis, P.A. Tarantili, and A.G. Andreopoulos Polymers for use in controlled release system: the effect of surfactants on their swelling properties J. Biomater. Appl. 15 2000 65 77
29. P.C. Wu, Y. Obata, M. Fujikawa, C.J. Li, K. Higashiyama, and K. Takayama Simultaneous optimization based on artificial neural networks in ketoprofen hydrol formula containing o-ethyl-3-butylcyclohexanol as percutaneous absorption enhancer J. Pharm. Sci. 90 2001 1004 1014
30. S. Zuleger, and B.C. Lippold Polymer particle erosion controlling drug release I. Factors influencing drug release and characterization of the release mechanism Int. J. Pharm. 217 2001 139 152