Docking study of ligands into the colchicine binding site of tubulin

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 19, Issue 6, 2004, Pages 541-547

  Farce, Amaury ^a   Loge, Cedric ^a   Gallet, Sebastien ^a   Lebegue, Nicolas ^a   Carato, Pascal ^a   Chavatte, Philippe ^a   Berthelot, Pascal ^a   Lesieur, Daniel ^a  

^a UNIV LILLE   (France)

Author keywords

Antimitotic agents; Binding site; Cancer; Colchicine; Docking; Tubulin

Indexed keywords

ALPHA TUBULIN; ANTIMITOTIC AGENT; ANTINEOPLASTIC AGENT; BENZOPYRIDOTHIADIAZEPINE DERIVATIVE; BETA TUBULIN; BP 38A; BP 38B; COLCHICINE; COMBRESTATIN DERIVATIVE; DIMER; DOCETAXEL; EPOTHILONE DERIVATIVE; ER 34410; N [2 [(4 HYDROXYPHENYL)AMINO] 3 PYRIDINYL] 4 METHOXYBENZENESULFONAMIDE; NF 402A; NF 402B; OXATHIAZEPINE DERIVATIVE; PACLITAXEL; TUBULIN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL DEATH; CONTROLLED STUDY; DRUG BINDING SITE; DRUG CLASSIFICATION; DRUG CYTOTOXICITY; DRUG STRUCTURE; LIGAND BINDING; MICROTUBULE ASSEMBLY; MITOSIS INHIBITION; MITOSIS SPINDLE; MOLECULAR INTERACTION; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIMITOTIC AGENTS; BINDING SITES; CELL LINE, TUMOR; COLCHICINE; HYDROGEN BONDING; LIGANDS; MICE; MOLECULAR STRUCTURE; PROTEIN CONFORMATION; PROTEIN STRUCTURE, TERTIARY; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; STRUCTURE-ACTIVITY RELATIONSHIP; TUBULIN;

EID: 11244309063     PISSN: 14756366     EISSN: None     Source Type: Journal    
DOI: 10.1080/14756360412331280545     Document Type: Article

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