Inhibition of ATP-sensitive K+ channels by taurine through a benzamido-binding site on sulfonylurea receptor 1

Biochemical Pharmacology

Volumn 67, Issue 6, 2004, Pages 1089-1096

  Park, Eun Jee ^a   Bae, Jae Hoon ^b   Kim, So Yeon ^b   Lim, Jeong Geun ^a   Baek, Won Ki ^a   Kwon, Taeg Kyu ^a   Suh, Seong Il ^a   Park, Jong Wook ^a   Lee, In Kyu ^a   Ashcroft, Frances M ^c   Song, Dae Kyu ^b  

^a Keimyung University   (South Korea)

^b Department of Physiology ^*  (South Korea)

^c UNIVERSITY OF OXFORD   (United Kingdom)

Author keywords

Ca2+ c; ATP sensitive potassium channel; Cytosolic free Ca2+ concentration; H; Half maximal concentration for inhibition; Hill coefficient; IC50; KATP channel; Open probability; Po; SUR

Indexed keywords

ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATASE (POTASSIUM); ADENOSINE TRIPHOSPHATE; CALCIUM ION; COLLAGENASE; GLIBENCLAMIDE; GLICLAZIDE; MAGNESIUM; POTASSIUM CHANNEL; SULFONYLUREA RECEPTOR; SULFONYLUREA RECEPTOR 1; TAURINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG BINDING SITE; DRUG MECHANISM; FEMALE; FLUOROMETRY; INSULIN RELEASE; MALE; MEMBRANE POTENTIAL; NONHUMAN; NUCLEOTIDE SEQUENCE; OOCYTE; PANCREAS ISLET BETA CELL; PATCH CLAMP; POTASSIUM CURRENT; PRIORITY JOURNAL; RADIOIMMUNOASSAY; RAT; XENOPUS LAEVIS;

ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATE; ANIMALS; BINDING SITES; DRUG INTERACTIONS; GLYBURIDE; INSULIN; ISLETS OF LANGERHANS; MALE; MEMBRANE PROTEINS; POTASSIUM CHANNELS; POTASSIUM CHANNELS, INWARDLY RECTIFYING; PROTEIN SUBUNITS; RATS; RATS, SPRAGUE-DAWLEY; SULFONYLUREA COMPOUNDS; TAURINE;

EID: 10744226060     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2003.11.003     Document Type: Article

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