2,3-Diaminopyridine bradykinin B1 receptor antagonists

Journal of Medicinal Chemistry

Volumn 47, Issue 26, 2004, Pages 6439-6442

  Kuduk, Scott D ^a   Ng, Christina ^a   Feng, Dong Mei ^a   Wai, Jenny M C ^a   Chang, Raymond S L ^a   Harrell, Charles M ^a   Murphy, Kathy L ^a   Ransom, Richard W ^a   Reiss, Duane ^a   Ivarsson, Magnus ^b   Mason, Glenn ^b   Boyce, Susan ^b   Tang, Cuyue ^a   Prueksaritanont, Thomayant ^a   Freidinger, Roger M ^a   Pettibone, Douglas J ^a   Bock, Mark G ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

^b NEUROSCIENCE RESEARCH CENTRE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2,3 DIAMINOPYRIDINE DERIVATIVE; BRADYKININ B1 RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING AFFINITY; CHRONIC PAIN; CONTROLLED STUDY; DRUG BINDING; DRUG EFFICACY; DRUG STRUCTURE; DRUG SYNTHESIS; IN VIVO STUDY; INFLAMMATION; NONHUMAN; RABBIT; SPECIES DIFFERENCE;

AMINOPYRIDINES; ANALGESICS; ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; DOGS; HALF-LIFE; INFLAMMATION; PAIN MEASUREMENT; RABBITS; RATS; RECEPTOR, BRADYKININ B1; SPECIES SPECIFICITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 10644255580     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm049394l     Document Type: Article

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