Development of Novel Assays for Proteolytic Enzymes Using Rhodamine-Based Fluorogenic Substrates

Journal of Biomolecular Screening

Volumn 7, Issue 6, 2002, Pages 531-540

  Grant, Stephan K ^a,b   Sklar, Joseph G ^a,b,c   Cummings, Richard T ^a,d  

^a Department of Human and Animal Infectious Disease Research ^*  (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

^c PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

^d PRINCETON UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BACLOFEN; CYTOSOL AMINOPEPTIDASE; DIPEPTIDYL PEPTIDASE; DRUG DERIVATIVE; FLUORESCENT DYE; PENTAMIDINE; PEPTIDE; PHACLOFEN; PROTEINASE; PROTEINASE INHIBITOR; RHODAMINE;

ARTICLE; BIOASSAY; CHEMISTRY; COMBINATORIAL CHEMISTRY; DRUG ANTAGONISM; ENZYME SPECIFICITY; IC 50; METABOLISM; METHODOLOGY;

BACLOFEN; BIOLOGICAL ASSAY; COMBINATORIAL CHEMISTRY TECHNIQUES; DIPEPTIDYL PEPTIDASES; ENDOPEPTIDASES; FLUORESCENT DYES; INHIBITORY CONCENTRATION 50; LEUCYL AMINOPEPTIDASE; PENTAMIDINE; PEPTIDES; PROTEASE INHIBITORS; RHODAMINES; SUBSTRATE SPECIFICITY;

EID: 0642378377     PISSN: 10870571     EISSN: None     Source Type: Journal    
DOI: 10.1177/1087057102238627     Document Type: Article

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