Synthesis of pyrrolopyrimidine CRF-R1 antagonists containing a tricyclic core via an intramolecular heck reaction

Heterocycles

Volumn 62, Issue , 2004, Pages 191-195

  Dyck, Brian ^a   McCarthy, James R ^a,b  

^a NEUROCRINE BIOSCIENCES INC   (United States)

^b ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CORTICOTROPIN RELEASING FACTOR RECEPTOR; CORTICOTROPIN RELEASING FACTOR RECEPTOR 1; PALLADIUM; PYRROLOPYRIMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL MODIFICATION; CHEMICAL REACTION; CYCLIZATION; DRUG STRUCTURE; DRUG SYNTHESIS; PHARMACEUTICS; STEREOCHEMISTRY;

EID: 0347090301     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-03-S(P)41     Document Type: Article

References (14)

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13. The hCRF-R1 binding assay was performed as previously described.2
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