Syntheses and receptor-binding studies of derivatives of the opioid antagonist naltrexone

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 2, 2004, Pages 417-421

  Uwai, Koji ^a   Uchiyama, Hiroko ^a   Sakurada, Shinobu ^a   Kabuto, Chizuko ^b   Takeshita, Mitsuhiro ^a  

^a TOHOKU PHARMACEUTICAL UNIVERSITY   (Japan)

^b TOHOKU UNIVERSITY   (Japan)

Author keywords

Analgesia; Naltrexone derivatives; Opioid; Receptor binding assay

Indexed keywords

HYDROXYL GROUP; MU OPIATE RECEPTOR; NALTREXONE DERIVATIVE; OPIATE ANTAGONIST;

ARTICLE; BINDING AFFINITY; DRUG ACTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; OXYGENATION; RECEPTOR BINDING;

EID: 0346059511     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2003.10.039     Document Type: Article

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