메뉴 건너뛰기




Volumn 20, Issue 11, 1999, Pages 1311-1319

High-affinity binding of urocortin and astressin but not CRF to G protein-uncoupled CRFR1

Author keywords

5' cyclic monophosphate); Astressin; cAMP (adenosine 3'; CD (circular dichroism); CRF (corticotropin releasing factor); CRFR1 (CRF receptor: type 1); G protein coupling; GTP S (guanosine 5' O (3 thiotriphosphate)); RPHPLC (reverse phase HPLC); Ucn (urocortin)

Indexed keywords

ASTRESSIN; CORTICOTROPIN RELEASING FACTOR ANTAGONIST; CORTICOTROPIN RELEASING FACTOR DERIVATIVE; CORTICOTROPIN RELEASING FACTOR RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; MESSENGER RNA; NEUROPEPTIDE; UNCLASSIFIED DRUG; UROCORTIN;

EID: 0344560606     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(99)00136-9     Document Type: Article
Times cited : (21)

References (46)
  • 1
    • 0030229898 scopus 로고    scopus 로고
    • Neurobiology of corticotropin releasing factor (CRF) receptors and CRF-binding protein: Implications for the treatment of CNS disorders
    • Behan D.P., Grigoriadis D.E., Lovenberg T., Chalmers D., Heinrichs S., Liaw C., De Souza E.B. Neurobiology of corticotropin releasing factor (CRF) receptors and CRF-binding protein implications for the treatment of CNS disorders . Mol Psychiatry. 1:1996;265-277.
    • (1996) Mol Psychiatry , vol.1 , pp. 265-277
    • Behan, D.P.1    Grigoriadis, D.E.2    Lovenberg, T.3    Chalmers, D.4    Heinrichs, S.5    Liaw, C.6    De Souza, E.B.7
  • 3
    • 0029786101 scopus 로고    scopus 로고
    • A single-point slight alteration set as a tool for structure-activity relationship studies of ovine corticotropin releasing factor
    • Beyermann M., Fechner K., Furkert J., Krause E., Bienert M. A single-point slight alteration set as a tool for structure-activity relationship studies of ovine corticotropin releasing factor. J Med Chem. 39:1996;3324-3330.
    • (1996) J Med Chem , vol.39 , pp. 3324-3330
    • Beyermann, M.1    Fechner, K.2    Furkert, J.3    Krause, E.4    Bienert, M.5
  • 4
    • 0027716529 scopus 로고
    • Identification of a seven transmembrane helix receptor for corticotropin-releasing factor and sauvagine in mammalian brain
    • Chang C.P., Pearse R.V. II, O'Connell S., Rosenfeld M.G. Identification of a seven transmembrane helix receptor for corticotropin-releasing factor and sauvagine in mammalian brain. Neuron. 11:1993;1187-1195.
    • (1993) Neuron , vol.11 , pp. 1187-1195
    • Chang, C.P.1    Pearse R.V. II2    O'Connell, S.3    Rosenfeld, M.G.4
  • 5
    • 0027489208 scopus 로고
    • Expression cloning of a human corticotropin-releasing-factor receptor
    • Chen R., Lewis K.A., Perrin M.H., Vale W.W. Expression cloning of a human corticotropin-releasing-factor receptor. Proc Natl Acad Sci USA. 90:1993;8967-8971.
    • (1993) Proc Natl Acad Sci USA , vol.90 , pp. 8967-8971
    • Chen, R.1    Lewis, K.A.2    Perrin, M.H.3    Vale, W.W.4
  • 6
    • 0015967881 scopus 로고
    • Conformational parameters for amino acids in helical, β-sheet, and random coil regions calculated from proteins
    • Chou P.Y., Fasman G.D. Conformational parameters for amino acids in helical, β-sheet, and random coil regions calculated from proteins. Biochemistry. 13:1974;211-245.
    • (1974) Biochemistry , vol.13 , pp. 211-245
    • Chou, P.Y.1    Fasman, G.D.2
  • 7
    • 0030963837 scopus 로고    scopus 로고
    • Identification of two corticotropin-releasing factor receptors from xenopus laevis with high ligand selectivity: Unusual pharmacology of the type 1 receptor
    • Dautzenberg F.M., Dietrich K., Palchaudhuri M.R., Spiess J. Identification of two corticotropin-releasing factor receptors from xenopus laevis with high ligand selectivity unusual pharmacology of the type 1 receptor . J Neurochem. 69:1997;1640-1649.
    • (1997) J Neurochem , vol.69 , pp. 1640-1649
    • Dautzenberg, F.M.1    Dietrich, K.2    Palchaudhuri, M.R.3    Spiess, J.4
  • 8
    • 0021958530 scopus 로고
    • Corticotropin-releasing factor receptors in human pituitary gland: Autoradiographic localization
    • De Souza E.B., Perrin M.H., Whithouse P.J., Rivier J., Vale W.W., Kuhar M.J. Corticotropin-releasing factor receptors in human pituitary gland autoradiographic localization . Neuroendocrinol. 40:1985;419-422.
    • (1985) Neuroendocrinol , vol.40 , pp. 419-422
    • De Souza, E.B.1    Perrin, M.H.2    Whithouse, P.J.3    Rivier, J.4    Vale, W.W.5    Kuhar, M.J.6
  • 11
    • 0008228191 scopus 로고    scopus 로고
    • The C terminus ends of secretin and VIP interact with the N-terminal domains of their receptors
    • Gourlet P., Vilardaga J.P., De Neef P., Waelbroek M., Vandermeers A., Robberecht P. The C terminus ends of secretin and VIP interact with the N-terminal domains of their receptors. Peptides. 17:1996;825-829.
    • (1996) Peptides , vol.17 , pp. 825-829
    • Gourlet, P.1    Vilardaga, J.P.2    De Neef, P.3    Waelbroek, M.4    Vandermeers, A.5    Robberecht, P.6
  • 14
    • 0027283546 scopus 로고
    • Partial agonists, full agonists, antagonists: Dilemmas of definition
    • Hoyer D., Boddecke H.W.G.M. Partial agonists, full agonists, antagonists dilemmas of definition . Trends Pharmacol Sci. 14:1993;270-275.
    • (1993) Trends Pharmacol Sci , vol.14 , pp. 270-275
    • Hoyer, D.1    Boddecke, H.W.G.M.2
  • 16
    • 0031434924 scopus 로고    scopus 로고
    • Differences between natural and recombinant G protein-coupled receptor systems with varying receptor/G protein stoichiometry
    • Kenakin T. Differences between natural and recombinant G protein-coupled receptor systems with varying receptor/G protein stoichiometry. Trends Pharmacol Sci. 18:1997;456-464.
    • (1997) Trends Pharmacol Sci , vol.18 , pp. 456-464
    • Kenakin, T.1
  • 17
    • 0028800724 scopus 로고
    • A sauvagine/corticotropin-releasing factor receptor expressed in heart and skeletal muscle
    • Kishimoto T., Pearse R.V. II, Lin C.R., Rosenfeld M.G. A sauvagine/corticotropin-releasing factor receptor expressed in heart and skeletal muscle. Proc Natl Acad Sci USA. 92:1995;1108-1112.
    • (1995) Proc Natl Acad Sci USA , vol.92 , pp. 1108-1112
    • Kishimoto, T.1    Pearse R.V. II2    Lin, C.R.3    Rosenfeld, M.G.4
  • 19
    • 0029060237 scopus 로고
    • Location of an amphipathic α-helix in peptides by using reversed-phase HPLC retention behavior of D-amino acid analogs
    • Krause E., Beyermann M., Dathe M., Rothemund S., Bienert M. Location of an amphipathic α-helix in peptides by using reversed-phase HPLC retention behavior of D-amino acid analogs. Anal Chem. 67:1995;252-258.
    • (1995) Anal Chem , vol.67 , pp. 252-258
    • Krause, E.1    Beyermann, M.2    Dathe, M.3    Rothemund, S.4    Bienert, M.5
  • 20
    • 0030731863 scopus 로고    scopus 로고
    • Localization of agonist- And antagonist-binding domains of human corticotropin-releasing factor receptors
    • Liaw C.W., Grigoriadis D.E., Lorang M.T., De Souza E.B., Maki R.A. Localization of agonist- and antagonist-binding domains of human corticotropin-releasing factor receptors. Mol Endocrinol. 11:1997;2048-2053.
    • (1997) Mol Endocrinol , vol.11 , pp. 2048-2053
    • Liaw, C.W.1    Grigoriadis, D.E.2    Lorang, M.T.3    De Souza, E.B.4    Maki, R.A.5
  • 22
    • 0017280145 scopus 로고
    • An agonist-specific effect of guanine-nucleotides on binding to the beta adrenergic receptor
    • Maguire M.E., Van Arsdale P.M., Gilman A.G. An agonist-specific effect of guanine-nucleotides on binding to the beta adrenergic receptor. Mol Pharmacol. 12:1976;335-339.
    • (1976) Mol Pharmacol , vol.12 , pp. 335-339
    • Maguire, M.E.1    Van Arsdale, P.M.2    Gilman, A.G.3
  • 25
    • 0032559181 scopus 로고    scopus 로고
    • Distribution and concentration of urocortin, and effect of adrenalectomy on its content in rat hypothalamus
    • Oki Y., Iwabuchi M., Masuzawa M., Watanabe F., Ozawa M., Iino K., Yoshimi T. Distribution and concentration of urocortin, and effect of adrenalectomy on its content in rat hypothalamus. Life Sci. 62:1998;807-812.
    • (1998) Life Sci , vol.62 , pp. 807-812
    • Oki, Y.1    Iwabuchi, M.2    Masuzawa, M.3    Watanabe, F.4    Ozawa, M.5    Iino, K.6    Yoshimi, T.7
  • 26
    • 0343580125 scopus 로고
    • Structural homology of corticotropin-releasing factor, sauvagine, and urotensin I: Circular dichroism and prediction studies
    • Pallai P.V., Mabilla M., Goodman M., Vale W.W., Rivier J. Structural homology of corticotropin-releasing factor, sauvagine, and urotensin I circular dichroism and prediction studies . Proc Natl Acad Sci USA. 80:1983;6770-6774.
    • (1983) Proc Natl Acad Sci USA , vol.80 , pp. 6770-6774
    • Pallai, P.V.1    Mabilla, M.2    Goodman, M.3    Vale, W.W.4    Rivier, J.5
  • 27
    • 0022446474 scopus 로고
    • Corticotropin-releasing factor binding to the anterior pituitary receptor is modulated by divalent cations and guanyl nucleotides
    • Perrin M.H., Haas Y., Rivier J.E., Vale W.W. Corticotropin-releasing factor binding to the anterior pituitary receptor is modulated by divalent cations and guanyl nucleotides. Endocrinology. 118:1986;1171-1179.
    • (1986) Endocrinology , vol.118 , pp. 1171-1179
    • Perrin, M.H.1    Haas, Y.2    Rivier, J.E.3    Vale, W.W.4
  • 28
    • 0027131369 scopus 로고
    • Cloning and functional expression of a rat brain corticotropin releasing factor (CRF) receptor
    • Perrin M.H., Donaldson C.J., Chen R., Lewis K.A., Vale W.W. Cloning and functional expression of a rat brain corticotropin releasing factor (CRF) receptor. Endocrinology. 133:1993;3058-3061.
    • (1993) Endocrinology , vol.133 , pp. 3058-3061
    • Perrin, M.H.1    Donaldson, C.J.2    Chen, R.3    Lewis, K.A.4    Vale, W.W.5
  • 30
    • 0031764213 scopus 로고    scopus 로고
    • The first extracellular domain of corticotropin releasing factor-R1 contains major binding determinants for urocortin and astressin
    • Perrin M.H., Sutton S., Bain D.L., Berggren W.T., Vale W.W. The first extracellular domain of corticotropin releasing factor-R1 contains major binding determinants for urocortin and astressin. Endocrinology. 139:1998;566-570.
    • (1998) Endocrinology , vol.139 , pp. 566-570
    • Perrin, M.H.1    Sutton, S.2    Bain, D.L.3    Berggren, W.T.4    Vale, W.W.5
  • 32
    • 0020176542 scopus 로고
    • A constrained regularization method for inverting data represented by linear algebraic or integral equations
    • Provencher S.W. A constrained regularization method for inverting data represented by linear algebraic or integral equations. Comput Phys Commun. 27:1982;213-227.
    • (1982) Comput Phys Commun , vol.27 , pp. 213-227
    • Provencher, S.W.1
  • 33
    • 0027484160 scopus 로고
    • Single point D-substituted corticotropin-releasing factor analogues: Effects on potency and physicochemical characterization
    • Rivier J., Rivier C., Galyean R., Miranda A., Miller C., Craig A.G., Yamamoto G., Brown M., Vale W.W. Single point D-substituted corticotropin-releasing factor analogues effects on potency and physicochemical characterization . J Med Chem. 36:1993;2851-2859.
    • (1993) J Med Chem , vol.36 , pp. 2851-2859
    • Rivier, J.1    Rivier, C.2    Galyean, R.3    Miranda, A.4    Miller, C.5    Craig, A.G.6    Yamamoto, G.7    Brown, M.8    Vale, W.W.9
  • 35
    • 0029785198 scopus 로고    scopus 로고
    • Synthesis and characterization of a photoactivatable analog of corticotropin-releasing factor for specific receptor labeling
    • Rühmann A., Köpke A.K.E., Dautzenberg F.M., Spiess J. Synthesis and characterization of a photoactivatable analog of corticotropin-releasing factor for specific receptor labeling. Proc Natl Acad Sci USA. 93:1996;10609-10613.
    • (1996) Proc Natl Acad Sci USA , vol.93 , pp. 10609-10613
    • Rühmann, A.1    Köpke, A.K.E.2    Dautzenberg, F.M.3    Spiess, J.4
  • 36
    • 0032417612 scopus 로고    scopus 로고
    • Structural requirements for peptidic antagonists of the corticotropin-releasing factor receptor (CRFR): Development of CRFR2β-selective antisauvagine-30
    • Rühmann A., Bonk I., Lin C.R., Rosenfeld M.G., Spiess J. Structural requirements for peptidic antagonists of the corticotropin-releasing factor receptor (CRFR) development of CRFR2β-selective antisauvagine-30 . Proc Natl Acad Sci USA. 95:1998;15264-15269.
    • (1998) Proc Natl Acad Sci USA , vol.95 , pp. 15264-15269
    • Rühmann, A.1    Bonk, I.2    Lin, C.R.3    Rosenfeld, M.G.4    Spiess, J.5
  • 38
    • 0033555673 scopus 로고    scopus 로고
    • The role of the fourth extracellular domain of the rat corticotropin-releasing factor receptor type 1 in ligand binding
    • Sydow S., Flaccus A., Fischer A., Spiess J. The role of the fourth extracellular domain of the rat corticotropin-releasing factor receptor type 1 in ligand binding. Eur J Biochem. 259:1999;55-62.
    • (1999) Eur J Biochem , vol.259 , pp. 55-62
    • Sydow, S.1    Flaccus, A.2    Fischer, A.3    Spiess, J.4
  • 39
    • 0032892757 scopus 로고    scopus 로고
    • Urocortin is not a significant regulator of intermittent electrofootshock-induced adrenocorticotropin secretion in the intact male rat
    • Turnbull A.V., Vaughan J., Rivier J.E., Vale W.W., Rivier C. Urocortin is not a significant regulator of intermittent electrofootshock-induced adrenocorticotropin secretion in the intact male rat. Endocrinology. 140:1999;71-78.
    • (1999) Endocrinology , vol.140 , pp. 71-78
    • Turnbull, A.V.1    Vaughan, J.2    Rivier, J.E.3    Vale, W.W.4    Rivier, C.5
  • 40
    • 0030903884 scopus 로고    scopus 로고
    • A new functional isoform of the human CRF2 receptor for corticotropin-releasing factor
    • Valdenaire O., Giller T., Breu V., Gottowik J., Kilpatrick G. A new functional isoform of the human CRF2 receptor for corticotropin-releasing factor. Biochim Biophys Acta. 1352:1997;129-132.
    • (1997) Biochim Biophys Acta , vol.1352 , pp. 129-132
    • Valdenaire, O.1    Giller, T.2    Breu, V.3    Gottowik, J.4    Kilpatrick, G.5
  • 41
    • 0019782980 scopus 로고
    • Characterization of a 41 residue ovine hypothalamic peptide that stimulates secretion of corticotropin and β-endorphin
    • Vale W., Spiess J., Rivier C., Rivier J. Characterization of a 41 residue ovine hypothalamic peptide that stimulates secretion of corticotropin and β-endorphin. Science. 213:1981;1394-1397.
    • (1981) Science , vol.213 , pp. 1394-1397
    • Vale, W.1    Spiess, J.2    Rivier, C.3    Rivier, J.4
  • 45
    • 0030801196 scopus 로고    scopus 로고
    • The C terminal part of VIP is important for receptor binding and activation, as evidenced by chimeric constructs of VIP/secretin
    • Wulff B., Møller Knudsen S., Adelhorst K., Fahrenkrug J. The C terminal part of VIP is important for receptor binding and activation, as evidenced by chimeric constructs of VIP/secretin. FEBS Lett. 413:1997;405-408.
    • (1997) FEBS Lett , vol.413 , pp. 405-408
    • Wulff, B.1    Møller Knudsen, S.2    Adelhorst, K.3    Fahrenkrug, J.4
  • 46
    • 9044254926 scopus 로고    scopus 로고
    • Molecular cloning of a type A chicken corticotropin-releasing factor receptor with high affinity for urotensin I
    • Yu J., Xie L.Y., Abou-Samra A.B. Molecular cloning of a type A chicken corticotropin-releasing factor receptor with high affinity for urotensin I. Endocrinology. 137:1996;192-197.
    • (1996) Endocrinology , vol.137 , pp. 192-197
    • Yu, J.1    Xie, L.Y.2    Abou-Samra, A.B.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.