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Petersen, P.J., Jacobus, N.V., Weiss, W.J., Sum, P.E., Testa, R.T. In vitro and in vivo antibacterial activities of a novel glycylcycline, the 9-t-butylglycylamido derivative of minocycline (GAR-936). Antimicrob Agents Chemother 1999, 43: 738-44.
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In vitro activities of the glycylcycline GAR-936 against Gram-positive bacteria
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Boucher, H.W., Wennersten, C.B., Eliopoulos, G.M. In vitro activities of the glycylcycline GAR-936 against Gram-positive bacteria. Antimicrob Agents Chemother 2000, 44: 2225-9.
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In vitro activity of GAR-936 against vancomycin-resistant enterococci, methicillin-resistant Staphylococcus aureus and penicillin-resistant Streptococcus pneumoniae
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Patel, R., Rouse, M., Piper, K., Steckelberg, J. In vitro activity of GAR-936 against vancomycin-resistant enterococci, methicillin-resistant Staphylococcus aureus and penicillin-resistant Streptococcus pneumoniae. Diagn Microbiol Infect Dis 2000, 38: 177-9.
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Patel, R.1
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Antipneumococcal activities of GAR-936 (a new glycylcycline) compared to those of nine other agents against penicillin-susceptible and -resistant pneumococci
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Hoellman, D.B., Pankuch, G.A., Jacobs, M.R., Appelbaum, P.C. Antipneumococcal activities of GAR-936 (a new glycylcycline) compared to those of nine other agents against penicillin-susceptible and -resistant pneumococci. Antimicrob Agents Chemother 2000, 44: 1085-8.
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Antimicrobial activity and spectrum of the new glycylcycline, GAR-936 tested against 1,203 recent clinical bacterial isolates
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Gales, A.C., Jones, R.N. Antimicrobial activity and spectrum of the new glycylcycline, GAR-936 tested against 1,203 recent clinical bacterial isolates. Diagn Microbiol Infect Dis 2000, 36: 19-36.
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In-vitro susceptibility of anaerobic bacteria to GAR-936, a new glycylcycline
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Edlund, C., Nord, C. In-vitro susceptibility of anaerobic bacteria to GAR-936, a new glycylcycline. Clin Microbiol Infect 2000; 6: 159-163.
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Edlund, C.1
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10
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0033807573
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Comparative in vitro activities of GAR-936 against aerobic and anaerobic animal and human bite wound pathogens
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Goldstein, E., Citron, D., Merriam, C., Warren, Y., Tyrrell, K. Comparative In vitro activities of GAR-936 against aerobic and anaerobic animal and human bite wound pathogens. Antimicrob Agents Chemother 2000, 44: 2747-51.
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Antimicrob Agents Chemother
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Goldstein, E.1
Citron, D.2
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Tyrrell, K.5
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11
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In vitro activity of GAR-936 against Chlamydia pneumoniae and Chlamydia trachomatis
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Roblin, P.M., Hammerschlag, M.R. In vitro activity of GAR-936 against Chlamydia pneumoniae and Chlamydia trachomatis. Int J Antimicrob Agents 2000, 16: 61-3.
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Roblin, P.M.1
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12
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0347115148
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The susceptibilities of human mycoplasmas to a new glycylcycline, GAR-936
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Sept 26-29, San Francisco, Abst F412
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Kenny, G.E., Cartwright, F.D. The susceptibilities of human mycoplasmas to a new glycylcycline, GAR-936. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F412.
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39th Intersci Conf Antimicrob Agents Chemother
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Kenny, G.E.1
Cartwright, F.D.2
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13
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0033818355
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Preclinical pharmacology of GAR-936, a novel glycylcycline antibacterial agent
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Projan, S. Preclinical pharmacology of GAR-936, a novel glycylcycline antibacterial agent. Pharmacotherapy 2000; 20(9, Part 2, Supp. S): 219S-23S.
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Projan, S.1
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14
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Therapeutic efficacy of GAR-936, a novel glycylcycline, in murine infections
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Sept 24-27, San Diego, Abst F-135
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Mikels, S.M., Lenoy, E., Allen, W., Compton, S., Weiss, W.J. Therapeutic efficacy of GAR-936, a novel glycylcycline, in murine infections. 38th Intersci Conf Antimicrob Agents Chemother (Sept 24-27, San Diego) 1998, Abst F-135.
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(1998)
38th Intersci Conf Antimicrob Agents Chemother
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Mikels, S.M.1
Lenoy, E.2
Allen, W.3
Compton, S.4
Weiss, W.J.5
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15
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0347115120
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In vivo activities of GAR-936 (GAR), gentamicin (GEN), piperacillin (PIP) alone and in combination in a murine model of Pseudomonas pneumonia
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Sept 26-29, San Francisco, Abst F414
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Mikels, S.M., Brown, A.S., Breden, L., Compton, S., Mitelman, S., Petersen, P.J., Weiss, W.J. In vivo activities of GAR-936 (GAR), gentamicin (GEN), piperacillin (PIP) alone and in combination in a murine model of Pseudomonas pneumonia. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F414.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Mikels, S.M.1
Brown, A.S.2
Breden, L.3
Compton, S.4
Mitelman, S.5
Petersen, P.J.6
Weiss, W.J.7
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16
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0034075749
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In vivo pharmacodynamic activities of two glycylcyclines (GAR-936 and WAY 152,288) against various Gram-positive and Gram-negative bacteria
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van Ogtrop, M.L., Andes, D., Stamstad, T.J., Conklin, B., Weiss, W.J., Craig, W.A., Vesga, O. In vivo pharmacodynamic activities of two glycylcyclines (GAR-936 and WAY 152,288) against various Gram-positive and Gram-negative bacteria. Antimicrob Agents Chemother 2000, 44: 943-9.
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Antimicrob Agents Chemother
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Van Ogtrop, M.L.1
Andes, D.2
Stamstad, T.J.3
Conklin, B.4
Weiss, W.J.5
Craig, W.A.6
Vesga, O.7
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17
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0033734720
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Therapeutic efficacy of GAR-936, a novel glycylcycline, in a rat model of experimental endocarditis
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Murphy, T., Deitz, J., Petersen, P., Mikels, S., Weiss, W. Therapeutic efficacy of GAR-936, a novel glycylcycline, in a rat model of experimental endocarditis. Antimicrob Agents Chemother 2000, 44: 3022-7.
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Antimicrob Agents Chemother
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, pp. 3022-3027
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Murphy, T.1
Deitz, J.2
Petersen, P.3
Mikels, S.4
Weiss, W.5
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18
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0347115119
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Activity and diffusion of GAR-936 in experimental enterococcal endocarditis
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Sept 26-29, San Francisco, Abst F415
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Lefort, A., Lafaurie, M., Saleh-Mghir, A., Garry, L., Peker, M.C., Le Guludec, D., Carbon, C., Fantin, B. Activity and diffusion of GAR-936 in experimental enterococcal endocarditis. 39th Intersci Coni Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F415.
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(1999)
39th Intersci Coni Antimicrob Agents Chemother
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Lefort, A.1
Lafaurie, M.2
Saleh-Mghir, A.3
Garry, L.4
Peker, M.C.5
Le Guludec, D.6
Carbon, C.7
Fantin, B.8
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19
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23844469695
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Comparative efficacy of GAR-936 (GAR), a novel glycylcycline, alone and in combination with vancomycin against highly penicillin-resistant Streptococcus pneumoniae (PRSP) experimental meningitis in rabbits
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Sept 17-20, Toronto, Abst B-868
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Fang, G.D., Weiss, W.J., Scheld, W.M. Comparative efficacy of GAR-936 (GAR), a novel glycylcycline, alone and in combination with vancomycin against highly penicillin-resistant Streptococcus pneumoniae (PRSP) experimental meningitis in rabbits. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst B-868.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
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Fang, G.D.1
Weiss, W.J.2
Scheld, W.M.3
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20
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23844436190
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Tissue distribution of GAR-936, a broad spectrum antibiotic in rats
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Sept 26-29, San Francisco, Abst F413
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Tombs, N.L. Tissue distribution of GAR-936, a broad spectrum antibiotic in rats. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F413.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Tombs, N.L.1
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21
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0002702892
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Pharmacokinetics (PK), safety and tolerability of GAR-936, a novel glycylcycline antibiotic, in healthy subjects
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Sept 26-29, San Francisco, Abst F416
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Muralidharan, G., Gesty, J., Mayer, P., Paty, I., Micalizzi, M., Speth, J., Wester, B., Mojaverian, P. Pharmacokinetics (PK), safety and tolerability of GAR-936, a novel glycylcycline antibiotic, in healthy subjects. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F416.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Muralidharan, G.1
Gesty, J.2
Mayer, P.3
Paty, I.4
Micalizzi, M.5
Speth, J.6
Wester, B.7
Mojaverian, P.8
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22
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0345853870
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The effects of age and gender on the pharmacokinetics, safety and tolerability of GAR-936, a novel glycylcycline antibiotic, in healthy subjects
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Sept 17-20, Toronto, Abst A-502
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Muralidharan, G., Mojaverian, P., Micalizzi, M., Speth, J., Tse, S., Stroshane, R., Getsy, J., Mayer, P. The effects of age and gender on the pharmacokinetics, safety and tolerability of GAR-936, a novel glycylcycline antibiotic, in healthy subjects. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst A-502.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
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Muralidharan, G.1
Mojaverian, P.2
Micalizzi, M.3
Speth, J.4
Tse, S.5
Stroshane, R.6
Getsy, J.7
Mayer, P.8
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25
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85037396262
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Mutations in the interdomain region of tetA(A) lead to glycylcycline-resistance in Salmonella isolates
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Sept 24-27, San Diego, Abst C-98
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Tuckman, M., Petersen, P.J., Projan, S.J. Mutations in the interdomain region of tetA(A) lead to glycylcycline-resistance in Salmonella isolates. 38th Intersci Conf Antimicrob Agents Chemother (Sept 24-27, San Diego) 1998, Abst C-98.
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(1998)
38th Intersci Conf Antimicrob Agents Chemother
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Tuckman, M.1
Petersen, P.J.2
Projan, S.J.3
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26
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0006314582
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The post-antibiotic effect and time-kill kinetics of the glycylcyclines, GAR-936 (TBG-MINO) and PAM-MINO
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Sept 24-27, San Diego, Abst F-132
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Petersen, P.J., Weiss, W.J., Labthavikul, P., Bradford, P.A. The post-antibiotic effect and time-kill kinetics of the glycylcyclines, GAR-936 (TBG-MINO) and PAM-MINO. 38th Intersci Conf Antimicrob Agents Chemother (Sept 24-27, San Diego) 1998, Abst F-132.
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(1998)
38th Intersci Conf Antimicrob Agents Chemother
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Petersen, P.J.1
Weiss, W.J.2
Labthavikul, P.3
Bradford, P.A.4
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27
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0008930343
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GAR-936, a novel glycylcycline, in the treatment of experimental endocarditis
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Sept 24-27, San Diego, Abst F-136
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Weiss, W.J., Murphy, T.M., Mikels, S.M., Clegg, J. GAR-936, a novel glycylcycline, in the treatment of experimental endocarditis. 38th Intersci Conf Antimicrob Agents Chemother (Sept 24-27, San Diego) 1998, Abst F-136.
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(1998)
38th Intersci Conf Antimicrob Agents Chemother
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Weiss, W.J.1
Murphy, T.M.2
Mikels, S.M.3
Clegg, J.4
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28
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0346484790
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In vitro activity of GAR-936 against Gram-positive bacteria
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Sept 26-29, San Francisco, Abst F406
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Boucher, H.W., Wennersten, C.B., Moellering, R.C., Eliopoulos, G.M. In vitro activity of GAR-936 against Gram-positive bacteria. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F406.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Boucher, H.W.1
Wennersten, C.B.2
Moellering, R.C.3
Eliopoulos, G.M.4
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29
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0037570407
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Antimicrobial activity of the novel glycylcycline GAP-936, tested against over 1000 recent clinical isolates including multiresistant Gram-positive cocci
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Sept 26-29, San Francisco, Abst F407
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Jones, R.N., Gales, A.C., Deshpande, L.M., Johnson, D.M., Biedenbach, D.J. Antimicrobial activity of the novel glycylcycline GAP-936, tested against over 1000 recent clinical isolates including multiresistant Gram-positive cocci. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F407.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Jones, R.N.1
Gales, A.C.2
Deshpande, L.M.3
Johnson, D.M.4
Biedenbach, D.J.5
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30
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0347115113
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In vitro activity of new glycylcycline, GAR 936 against methillicin-resistant and -susceptible Staphylococcus aureus isolated in North America
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Sept 26-29, San Francisco, Abst F408
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Mahalinggam, E., Trepeski, L., Pong-Porter, S., De Azavedo, J., Low, D.E., Kreiswirtn, B.N. In vitro activity of new glycylcycline, GAR 936 against methillicin-resistant and -susceptible Staphylococcus aureus isolated in North America. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F408.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Mahalinggam, E.1
Trepeski, L.2
Pong-Porter, S.3
De Azavedo, J.4
Low, D.E.5
Kreiswirtn, B.N.6
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31
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0347115116
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Antipneumococcal activity of GAR 936, a new glycylcycline, by agar dilution MIC
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Sept 26-29, San Francisco, Abst F409
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Hoellman, D.B., Jacobs, M.R., Appelbaum, P.C. Antipneumococcal activity of GAR 936, a new glycylcycline, by agar dilution MIC. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F409.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Hoellman, D.B.1
Jacobs, M.R.2
Appelbaum, P.C.3
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32
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0347115115
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Antipneumoccocal activity of GAR 936, a new glycylcycline, compared with seven compounds by broth dilution and time-kill
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Sept 26-29, San Francisco, Abst F410
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Pankuch, G.A., Jacobs, M.R., Appelbaum, P.C. Antipneumoccocal activity of GAR 936, a new glycylcycline, compared with seven compounds by broth dilution and time-kill. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F410.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Pankuch, G.A.1
Jacobs, M.R.2
Appelbaum, P.C.3
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33
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0345853869
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In vitro activity of anaerobic bacteria to GAR-936, a new glycylcycline
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Sept 26-29, San Francisco, Abst F411
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Hedberg, M., Nord, C.E. In vitro activity of anaerobic bacteria to GAR-936, a new glycylcycline. 39th Intersci Conf Antimicrob Agents Chemother (Sept 26-29, San Francisco) 1999, Abst F411.
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(1999)
39th Intersci Conf Antimicrob Agents Chemother
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Hedberg, M.1
Nord, C.E.2
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34
-
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0346484786
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Effect of in vitro test methodologies on the activity of the glycylcyclines against Streptococcus pneumoniae
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Sept 17-20, Toronto, Abst D-333
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Petersen, P.J., Rittenhouse, J.L., Sum, P.E., Bradford, P.A. Effect of in vitro test methodologies on the activity of the glycylcyclines against Streptococcus pneumoniae. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst D-333.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
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Petersen, P.J.1
Rittenhouse, J.L.2
Sum, P.E.3
Bradford, P.A.4
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35
-
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0347745406
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Comparative in vitro activity of GAR-936, a novel glycylglycine, against 422 strains of unususal aerobic and anaerobic bacteria isolated from infected bite wounds
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Sept 17-20, Toronto, Abst E-524
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Citron, D.M., Goldstein, E.J.C. Comparative in vitro activity of GAR-936, a novel glycylglycine, against 422 strains of unususal aerobic and anaerobic bacteria isolated from infected bite wounds. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst E-524.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
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Citron, D.M.1
Goldstein, E.J.C.2
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36
-
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0345853868
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In vitro susceptibility of adherent (biofilm) S. epidermidis clinical isolates to GAR-936 (GAR), minocycline (MINO) and vancomycin (VAN)
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Sept 17-20, Toronto, Abst E-525
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Labthavikul, P., Bradford, P.A. In vitro susceptibility of adherent (biofilm) S. epidermidis clinical isolates to GAR-936 (GAR), minocycline (MINO) and vancomycin (VAN). 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst E-525.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
-
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Labthavikul, P.1
Bradford, P.A.2
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37
-
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0347115109
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In vitro activity of GAR-936 against vancomycin resistant enterococci, methicillin-resistant Staphylococcus aureus, and penicillin-resistant pneumococci
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Sept 17-20, Toronto, Abst E-526
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Piper, K.E., Rouse, M.S., Wilson, W.R., Steckelberg, J.M., Patel, R. In vitro activity of GAR-936 against vancomycin resistant enterococci, methicillin-resistant Staphylococcus aureus, and penicillin-resistant pneumococci. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst E-526.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
-
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Piper, K.E.1
Rouse, M.S.2
Wilson, W.R.3
Steckelberg, J.M.4
Patel, R.5
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38
-
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0347115112
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Activities of GAR-936 alone and in combination versus multi-drug resistant Staphylococcus aureus and Enterococcus faecium
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Sept 17-20, Toronto, Abst E-532
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Mercier, R.C., Kennedy, C., Meadows, C. Activities of GAR-936 alone and in combination versus multi-drug resistant Staphylococcus aureus and Enterococcus faecium. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst E-532.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
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Mercier, R.C.1
Kennedy, C.2
Meadows, C.3
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39
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0347745408
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Pharmacodynamics of GAR 936 (GAR) in experimental endocarditis due to VanA-type Enterococcus faecium
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Sept 17-20, Toronto, Abst A-2256
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Lefort, A., Massias, L., Saleh-Mghir, A., Lafaurie, M., Garry, L., Carbon, C., Fantin, B. Pharmacodynamics of GAR 936 (GAR) in experimental endocarditis due to VanA-type Enterococcus faecium. 40th Intersci Conf Antimicrob Agents Chemother (Sept 17-20, Toronto) 2000, Abst A-2256.
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(2000)
40th Intersci Conf Antimicrob Agents Chemother
-
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Lefort, A.1
Massias, L.2
Saleh-Mghir, A.3
Lafaurie, M.4
Garry, L.5
Carbon, C.6
Fantin, B.7
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