4-Aminobicyclo[2.2.2]octanone Derivatives with Antiplasmodial and Antitrypanosomal Activities

Monatshefte fur Chemie

Volumn 134, Issue 10, 2003, Pages 1411-1420

  Seebacher, Werner ^a   Brun, Reto ^b   Saf, Robert ^c   Weis, Robert ^a  

^a UNIVERSITY OF GRAZ   (Austria)

^b SWISS TROPICAL AND PUBLIC HEALTH INSTITUTE   (Switzerland)

^c GRAZ UNIVERSITY OF TECHNOLOGY   (Austria)

Author keywords

Antiplasmodial activity; Antitrypanosomal activity; Bicyclo 2.2.2 octane derivatives; Oxidations; Reductions

Indexed keywords

4 (N OXIDODIMETHYLAMINO) 6,7 DIPHENYLBICYCLO[2.2.2]OCTAN 2 ONE; 4 (N OXIDOMORPHOLINO) 6,7 DIPHENYLBICYCLO[2.2.2]OCTAN 2 ONE; 4 (N OXIDOPIPERIDINO) 6,7 DIPHENYLBICYCLO[2.2.2]OCTAN 2 ONE; 4 (N OXIDOPYRROLIDINO) 6,7 DIPHENYLBICYCLO[2.2.2]OCTAN 2 ONE; 4 DIMETHYLAMINO 6,7 BIS(4 METHOXYPHENYL)BICYCLO[2.2.2]OCTAN 2 ONE; 4 DIMETHYLAMINO 6,7 DIPHENYLBICYCLO[2.2.2]OCTANE; 4 MORPHOLINO 6,7 DIPHENYLBICYCLO[2.2.2]OCTANE; 6,7 BIS(4 METHOXYPHENYL) 4 MORPHOLINOBICYCLO[2.2.2]OCTAN 2 ONE; 6,7 BIS(4 METHOXYPHENYL) 4 PIPERIDINOBICYCLO[2.2.2]OCTAN 2 ONE; 6,7 BIS(4 METHOXYPHENYL) 4 PYRROLIDINOBICYCLO[2.2.2]OCTAN 2 ONE; 6,7 DIPHENYL 4 PIPERIDINOBICYCLO[2.2.2]OCTANE; 6,7 DIPHENYL 4 PYRROLIDINOBICYCLO[2.2.2]OCTANE; ANTIMALARIAL AGENT; ANTITRYPANOSOMAL AGENT; BICYCLO COMPOUND; OCTANE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION; TRYPANOSOMA RHODESIENSE;

EID: 0141976650     PISSN: 00269247     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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