A catch-and-release strategy for the combinatorial synthesis of 4-acylamino-1,3-thiazoles as potential CDK5 inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 20, 2003, Pages 3491-3495

  Larsen, Scott D ^a   Stachew, Carl F ^a   Clare, Paula M ^a   Cubbage, Jerry W ^a   Leach, Karen L ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLIN A; CYCLIN DEPENDENT KINASE 2; CYCLIN DEPENDENT KINASE 5; CYCLIN DEPENDENT KINASE INHIBITOR; THIAZOLE DERIVATIVE;

ARTICLE; COMBINATORIAL CHEMISTRY; CONTROLLED DRUG RELEASE; CURTIUS REARRANGEMENT; DRUG RELEASE; DRUG SELECTIVITY; REGENERATION;

EID: 0141517081     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00726-1     Document Type: Article

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