Correlation between the affinity of flavonoids binding to the cytosolic site of Leishmania tropica multidrug transporter and their efficiency to revert parasite resistance to daunomycin

Biochemistry

Volumn 38, Issue 6, 1999, Pages 1736-1743

  Pérez Victoria, José M ^a   Chiquero, M Jesús ^a   Conseil, Gwenaëlle ^b   Dayan, Guila ^b   Pietro, Attilio Di ^b   Barron, Denis ^c   Castanys, Santiago ^a   Gamarro, Francisco ^a  

^a INSTITUTO DE PARASITOLOGÍA Y BIOMEDICINA LÓPEZ NEYRA   (Spain)

^b INSTITUT DE BIOLOGIE ET CHIMIE DES PROTÉINES   (France)

^c UNIVERSITÉ LYON 1   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ALLYL COMPOUND; CHROMONE DERIVATIVE; DAUNORUBICIN; FLAVANONE; FLAVONE; FLAVONOID; GENISTEIN; GLYCOPROTEIN P; HISTIDINE; ISOFLAVONE; ISOKAEMPFERIDE; MIFEPRISTONE; RHAMNOSE;

ARTICLE; BINDING AFFINITY; CYTOSOL; FLOW CYTOMETRY; HYDROPHOBICITY; LEISHMANIA TROPICA; MULTIDRUG RESISTANCE; NONHUMAN; PARASITE DEVELOPMENT; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN EXPRESSION; PROTEIN PURIFICATION;

ANIMALS; ATP-BINDING CASSETTE TRANSPORTERS; CELL LINE; CYTOSOL; DAUNORUBICIN; DRUG RESISTANCE, MULTIPLE; FLAVONOIDS; LEISHMANIA TROPICA; P-GLYCOPROTEIN; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; RECOMBINANT PROTEINS;

ESCHERICHIA COLI; LEISHMANIA TROPICA; PROTOZOA;

EID: 0039552151     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi982455v     Document Type: Article

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