2-Aminoethoxydiphenyl borate (2-APB) antagonises inositol 1,4,5-trisphosphate-induced calcium release, inhibits calcium pumps and has a use-dependent and slowly reversible action on store-operated calcium entry channels

Cell Calcium

Volumn 34, Issue 1, 2003, Pages 97-108

  Peppiatt, Claire M ^a   Collins, Tony J ^a   Mackenzie, Lauren ^a   Conway, Stuart J ^b   Holmes, Andrew B ^b   Bootman, Martin D ^a   Berridge, Michael J ^a   Seo, Jeong T ^a,c   Roderick, H Llewelyn ^a  

^a BABRAHAM INSTITUTE   (United Kingdom)

^b UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^c Yonsei University   (South Korea)

Author keywords

2 aminoethoxydiphenyl borate; Ca2+ signalling; InsP3

Indexed keywords

2 AMINOETHOXYDIPHENYLBORANE; ADENOSINE TRIPHOSPHATASE (CALCIUM); CALCIUM CHANNEL; CALCIUM ION; INOSITOL 1,4,5 TRISPHOSPHATE; INOSITOL 1,4,5 TRISPHOSPHATE RECEPTOR; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ARTICLE; CALCIUM CELL LEVEL; CALCIUM SIGNALING; CALCIUM TRANSPORT; CELL MEMBRANE DEPOLARIZATION; CONCENTRATION (PARAMETERS); CONCENTRATION RESPONSE; CONTROLLED STUDY; ELECTROSTIMULATION; HEART MUSCLE CELL; HELA CELL; HUMAN; HUMAN CELL; MITOCHONDRION; PRIORITY JOURNAL;

EID: 0038420824     PISSN: 01434160     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0143-4160(03)00026-5     Document Type: Article

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