Inhibition of the type 1 inositol 1,4,5-trisphosphate receptor by 2-aminoethoxydiphenylborate

Cellular Signalling

Volumn 14, Issue 11, 2002, Pages 955-960

  Bilmen, Jonathan G ^a   Michelangeli, Francesco ^a  

^a UNIVERSITY OF BIRMINGHAM   (United Kingdom)

Author keywords

2 APB; Ca2+; Ca2+ channels; Inhibition; Inositol 1,4,5 trisphosphate; InsP3 receptors

Indexed keywords

2 AMINOETHOXYDIPHENYLBORANE; ADENOSINE TRIPHOSPHATASE (CALCIUM); CALCIUM ION; INOSITOL 1,4,5 TRISPHOSPHATE RECEPTOR; RYANODINE RECEPTOR; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BRAIN MICROSOME; CALCIUM TRANSPORT; CEREBELLUM; COMPETITIVE INHIBITION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; DRUG MECHANISM; DRUG PENETRATION; DRUG POTENCY; ENZYME ACTIVITY; IC 50; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING;

ANIMALS; BINDING SITES; BORON COMPOUNDS; CALCIUM; CALCIUM CHANNEL BLOCKERS; CALCIUM CHANNELS; CALCIUM SIGNALING; CALCIUM-TRANSPORTING ATPASES; CELL MEMBRANE; DOSE-RESPONSE RELATIONSHIP, DRUG; EUKARYOTIC CELLS; INOSITOL 1,4,5-TRISPHOSPHATE; KINETICS; LIGANDS; MICROSOMES; RABBITS; RECEPTORS, CYTOPLASMIC AND NUCLEAR; SUBCELLULAR FRACTIONS; SWINE;

EID: 0036829060     PISSN: 08986568     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0898-6568(02)00042-6     Document Type: Article

References (28)

1. Berridge M.J., Bootman M.D., Lipp P. Nature. 395:1998;645-648.
2. Patel S., Joseph S.K., Thomas A.P. Cell Calcium. 25:1999;247-264.
3. Wojcikiewicz R.J. J. Biol. Chem. 270:1995;11678-11683.
4. Berridge M.J. Biochem. J. 312:1995;1-11.
5. Ma H.T., Venkatachalam K., Li H.S., Montell C., Kurosaki T., Patterson R.L., Gill D.L. J. Biol. Chem. 276:2001;18888-18896.
6. Gregory R.B., Rychkov G., Barritt G.J. Biochem. J. 354:2001;285-290.
7. Ma H.T., Patterson R.L., van Rossum D.B., Birnbaumer L., Mikoshiba K., Gill D.L. Science. 287:2000;1647-1651.
8. Maruyama T., Kanaji T., Nakade S., Kanno T., Mikoshiba K. J. Biochem. (Tokyo). 122:1997;498-505.
9. Longland C.L., Mezna M., Langel U., Hallbrink M., Soomets U., Wheatley M., Michelangeli F., Howl J. Cell Calcium. 24:1998;27-34.
10. Michelangeli F., Munkonge F.M. Anal. Biochem. 194:1991;231-236.
11. Michelangeli F. J. Fluoresc. 1:1991;203-206.
12. Michelangeli F. Cell Signal. 5:1993;33-39.
13. Mezna M., Michelangeli F. J. Biol. Chem. 270:1995;28097-28102.
14. Mezna M., Michelangeli F. Biochem. J. 325:1997;177-182.
15. Mezna M., Michelangeli F. J. Biol. Chem. 271:1996;31818-31823.
16. Tovey S.C., Dyer J.L., Godfrey R.E., Khan S.Z., Bilmen J.G., Mezna M., Michelangeli F. Pharmacol. Res. 42:2000;581-590.
17. Brown G.R., Sayers L.G., Kirk C.J., Michell R.H., Michelangeli F. Biochem. J. 282:1992;309-312.
18. Mezna M., Patchick T., Tovey S., Michelangeli F. Biochem. J. 314:1996;175-179.
19. Bilmen J.G., Khan S.Z., Javed M.U., Michelangeli F. Eur. J. Biochem. 268:2001;6318-6327.
20. Dyer J.L., Khan S.Z., Bilmen J.G., Hawtin S.R., Wheatley M., Javed M.U., Michelangeli F. Cell Calcium. 31:2002;45-52.
21. Tovey S.C., Longland C.L., Mezna M., Michelangeli F. Eur. J. Pharmacol. 354:1998;245-251.
22. Gafni J., Munsch J.A., Lam T.H., Catlin M.C., Costa L.G., Molinski T.F., Pessah I.N. Neuron. 19:1997;723-733.
23. Khan S.Z., Dyer J.L., Michelangeli F. Cell Signal. 13:2001;57-63.
24. Longland C.L., Dyer J.L., Michelangeli F. Eur. J. Pharmacol. 408:2000;219-225.
25. Sayers L.G., Michelangeli F. Biochem. Biophys. Res. Commun. 197:1993;1203-1208.
26. Sayers L.G., Michelangeli F. Biochim. Biophys. Acta. 1152:1993;177-183.
27. Pascual J.M., Shieh C.C., Kirsch G.E., Brown A.M. Biophys. J. 69:1995;428-434.
28. Missiaen L., Callewaert G., De Smedt H., Parys J.B. Cell Calcium. 29:2001;111-116.