Positive allosteric modulator of the human 5-HT2C receptor

Molecular Pharmacology

Volumn 64, Issue 1, 2003, Pages 78-84

  Im, Wha Bin ^a   Chio, Christopher L ^a   Alberts, Glen L ^a   Dinh, Dac M ^b  

^a Biology II/Neurobiology   (United States)

^b Discovery Technologies   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA GALACTOPYRANOSIDE; DOPAMINE 2 RECEPTOR; DOPAMINE 3 RECEPTOR; DOPAMINE RECEPTOR; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); INOSITOL 1,4,5 TRISPHOSPHATE; INOSITOL PHOSPHATE; MESULERGINE; PNU 170158; PNU 33078; PNU 43240; PNU 61734E; PNU 62344E; PNU 62804E; PNU 63502E; PNU 65287E; PNU 67220E; PNU 68607E; PNU 69176E; PNU 8750; PYRAN DERIVATIVE; PYRANOSIDE; QUINPIROLE; SEROTONIN 2A RECEPTOR; SEROTONIN 2B RECEPTOR; SEROTONIN 6 RECEPTOR; SEROTONIN 7 RECEPTOR; SEROTONIN RECEPTOR; UNCLASSIFIED DRUG;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; HUMAN; HUMAN CELL; MAMMAL CELL; MEMBRANE BINDING; MOLECULAR CLONING; OBESITY; PHENOTYPE; PRIORITY JOURNAL; RECEPTOR BINDING; RECEPTOR DENSITY; RECEPTOR UPREGULATION; SEROTONIN RELEASE; STRUCTURE ANALYSIS; SURFACE PROPERTY; TRANQUILIZING ACTIVITY;

ALLOSTERIC REGULATION; ANIMALS; CELLS, CULTURED; GALACTOSIDES; HUMANS; PIPERIDINES; RECEPTOR, SEROTONIN, 5-HT2C; RECEPTORS, SEROTONIN; SEROTONIN AGENTS;

EID: 0037899617     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.64.1.78     Document Type: Article

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