Identification of a series of CCK-2 receptor nonpeptide agonists: Sensitivity to stereochemistry and a receptor point mutation

Proceedings of the National Academy of Sciences of the United States of America

Volumn 100, Issue 9, 2003, Pages 5525-5530

  Kopin, Alan S ^a   McBride, Edward W ^a   Chen, Ci ^a   Freidinger, Roger M ^b   Chen, Duan ^c   Zhao, Chun Mei ^c   Beinborn, Martin ^a  

^a TUFTS MEDICAL CENTER   (United States)

^b MERCK RESEARCH LABORATORIES   (United States)

^c NORWEGIAN UNIVERSITY OF SCIENCE AND TECHNOLOGY   (Norway)

Author keywords

[No Author keywords available]

Indexed keywords

CHOLECYSTOKININ B RECEPTOR; CHOLECYSTOKININ RECEPTOR; PEPTIDE HORMONE; UNCLASSIFIED DRUG;

ARTICLE; CHIRALITY; DRUG SCREENING; ENANTIOMER; HUMAN; HUMAN CELL; LIGAND BINDING; PEPTIDE ANALYSIS; POINT MUTATION; PRIORITY JOURNAL; PROTEIN DOMAIN; RECEPTOR GENE; SECOND MESSENGER; STEREOCHEMISTRY; STOMACH MUCOSA; STRUCTURE ACTIVITY RELATION;

ANIMALS; BENZODIAZEPINONES; COS CELLS; HUMANS; MALE; MICE; MICE, INBRED C57BL; PHENYLUREA COMPOUNDS; POINT MUTATION; RECEPTOR, CHOLECYSTOKININ B; RECEPTORS, CHOLECYSTOKININ; RECOMBINANT PROTEINS; STEREOISOMERISM;

EID: 0037627265     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.0831223100     Document Type: Article

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