Minor modifications of a cholecystokinin-B/gastrin receptor non-peptide antagonist confer a broad spectrum of functional properties

Journal of Biological Chemistry

Volumn 273, Issue 23, 1998, Pages 14146-14151

  Beinborn, Martin ^a   Quinn, Suzanne M ^a   Kopin, Alan S ^a  

^a TUFTS UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2,3 DIHYDRO 1 METHYL 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL) 3 (3 METHYLPHENYL)UREA; 1 [2,3 DIHYDRO 1 (2' METHYLPHENACYL) 2 OXO 5 PHENYL 1H 1,4 BENZODIAZEPIN 3 YL] 3 (3 METHYLPHENYL)UREA; 1 [5 (3 AZABICYCLO[3.2.2]NON 3 YL) 2,3 DIHYDRO 1 METHYL 2 OXO 1H 1,4 BENZODIAZEPIN 3 YL] 3 (3 METHYLPHENYL)UREA; CHOLECYSTOKININ B RECEPTOR; GASTRIN ANTAGONIST; GASTRIN RECEPTOR; PD 135158; PD 136450; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; GENE MUTATION; HORMONE RECEPTOR INTERACTION; NONHUMAN; PRIORITY JOURNAL; PROTEIN MODIFICATION; RECEPTOR BINDING; SIGNAL TRANSDUCTION;

ANIMALS; BENZODIAZEPINES; BENZODIAZEPINONES; BINDING, COMPETITIVE; COS CELLS; HORMONE ANTAGONISTS; INOSITOL PHOSPHATES; MOLECULAR STRUCTURE; MUTATION; PEPTIDES; PHENYLUREA COMPOUNDS; RECEPTORS, CHOLECYSTOKININ; SIGNAL TRANSDUCTION; TRANSFECTION;

ANIMALIA;

EID: 0032486383     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.273.23.14146     Document Type: Article

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