A two-state model of antagonist-AT1 receptor interaction: Further support by binding studies at low temperature

Biochemical Pharmacology

Volumn 65, Issue 8, 2003, Pages 1339-1341

  Verheijen, Ilse ^a   De Backer, Jean Paul ^a   Vanderheyden, Patrick ^a   Vauquelin, Georges ^a  

^a VRIJE UNIVERSITEIT BRUSSEL   (Belgium)

Author keywords

Angiotensin II; Antagonist; AT1 receptor; CHO cells; Insurmountable; Two state model

Indexed keywords

2 BUTYL 4 CHLORO 1 [[2' (1H TETRAZOL 5 YL) 4 BIPHENYLYL]METHYL] 5 IMIDAZOLECARBOXYLIC ACID; ANGIOTENSIN 1 RECEPTOR; CANDESARTAN; IRBESARTAN; LIGAND; LOSARTAN;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BINDING ASSAY; COMPARATIVE STUDY; COMPUTER SIMULATION; CONTROLLED STUDY; DATA ANALYSIS; INCUBATION TIME; LOW TEMPERATURE; MOLECULAR MECHANICS; NONHUMAN; PRIORITY JOURNAL; REACTION ANALYSIS; THEORETICAL MODEL;

EID: 0037446264     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0006-2952(03)00073-X     Document Type: Article

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