Synthesis of some biginelli compounds in solvent medium using a photochemistry method

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 178, Issue 3, 2003, Pages 495-500

  Foroughifar, N ^a   Mobinikhaledi, A ^a   Fathinejad Jirandehi, H ^a  

^a ARAK UNIVERSITY   (Iran)

Author keywords

1,4 Dihydropyrimidine 2(1H) ones; DHPM; Photochemistry

Indexed keywords

5 ACYL 6 METHYL 4 (4 CHLOROPHENYL) 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE; 5 ACYL 6 METHYL 4 (4 DIMETHYLAMINOPHENYL) 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE; 5 ACYL 6 METHYL 4 PHENYL 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE; ALDEHYDE DERIVATIVE; BENZENE DERIVATIVE; ETHYL 6 METHYL 4 (2,5 DIMETHOXYPHENYL) 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 (4 CHLOROPHENYL) 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 (4 DIMETHYLAMINOPHENYL) 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 (4 METHYLPHENYL) 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 (4 NITROPHENYL) 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 PHENYL 2 OXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; ETHYL 6 METHYL 4 PHENYL 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; KETONE DERIVATIVE; PYRIMIDINE DERIVATIVE; SOLVENT; TERT BUTYL 6 METHYL 4 (4 CHLOROPHENYL) 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; TERT BUTYL 6 METHYL 4 (4 DIMETHYLAMINOPHENYL) 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; TERT BUTYL 6 METHYL 4 (4 METHOXYPHENYL) 2 THIOXO 1,2,3,4 TETRAHYDROPYRIMIDINE 5 CARBOXYLATE; THIOUREA DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CYCLOCONDENSATION; DRUG SYNTHESIS; IRRADIATION; PHOTOCHEMISTRY;

EID: 0037359859     PISSN: 10426507     EISSN: None     Source Type: Journal    
DOI: 10.1080/10426500307928     Document Type: Article

References (17)

1. P. Biginelli, Gazz. Chim. Itall., 23, 360 (1893).
2. C. O. Kappe, Tetrahedron, 49, 6937 (1993).
3. H. Cho et al., J. Med. Chem., 32, 2399 (1989).
4. S. K. Atwal et al., J. Med. Chem., 33, 2629 (1990).
5. G. C. Rovnyak et al., J. Med. Chem., 38, 119 (1995).
6. K. S. Atwal, B. N. Swanson, S. E. Unger, D. M. Floyed, S. Moreland, A. Hedberg, and B. C. O'Reilly, J. Med. Chem., 34, 806 (1991).
7. G. C. Rovnyak, K. S. Atwal, A. Hedberg, S. D. Kimball, S. Moreland, J. Z. Gougoutas, B. C. Oreilly, J. Schwartz, and F. M. Malley, J. Med. Chem., 35, 3254 (1992).
8. G. J. Grover, S. Dzwonczyk, D. M. McMullen, C. S. Normadinam, P. G. Sleph, and S. J. Moreland, Pharm., 26, 289 (1995).
9. C. O. Kappe and F. S. Falsone, Synlett., 718 (1998).
10. W. C. Wong, B. Lagu, D. Nagarathnam, M. R. Marzabadi, and C. Gluchowskj, PCT Int. Appl. WO 98 51, 311.
11. M. A. Bruce, G. S. Pointdexter, and G. Johnson, PCT Int. Appl. WO 98 33, 791.
12. C. O. Kappe, D. Kumar, and R. S. Varma, Synthesis, 1799-1803 (1999).
13. F. Bigi, S. Carloni, B. Frullanti, R. Maggi, and G. Sartori, Tetrahedron Lett., 40, 3465 (1999).
14. P. Wipf and A. Cunningham, Tetrahedron Lett., 36, 7819 (1995).
15. A. Studer, S. Hadida, R. Ferrito, S. Y. Kim, P. Jeger, P. Wipf, and D. P. Curran, Science, 275, 823 (1997).
16. A. Studer, P. Jeger, P. Wipf, and D. P. Curran, J. Org. Chem., 62, 2917 (1997).
17. B. C. O'Reilly and K. S. Atwal, Heterocycles, 26, 1185 (1987).