A comparative QSAR study on carbonic anhydrase and matrix metalloproteinase inhibition by sulfonylated amino acid hydroxamates

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 18, Issue 1, 2003, Pages 7-13

  Gupta, S P ^a   Maheswaran, V ^a   Pande, V ^a   Kumar, Dalip ^a  

^a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

Carbonic anhydrase inhibition; Clostridium histolyticum collagenase inhibition; Matrix metalloproteinase inhibition; Quantitative structure activity relationship (QSAR); Sulfonylated amino acid hydroxamates

Indexed keywords

AMINO ACID; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE INHIBITOR; CLOSTRIDIOPEPTIDASE A; COLLAGENASE INHIBITOR; GELATINASE B; HYDROXAMIC ACID DERIVATIVE; INTERSTITIAL COLLAGENASE; ISOENZYME; MATRIX METALLOPROTEINASE; MATRIX METALLOPROTEINASE INHIBITOR; STROMELYSIN 2; ZINC ION;

ARTICLE; CONTROLLED STUDY; DRUG POTENCY; ENZYME ACTIVITY; ENZYME ANALYSIS; ENZYME BINDING; ENZYME INHIBITION; ENZYME INHIBITOR INTERACTION; ENZYME REGULATION; ENZYME STRUCTURE; HYDROPHOBICITY; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

CARBONIC ANHYDRASE INHIBITORS; HYDROXAMIC ACIDS; MATRIX METALLOPROTEINASES; PROTEASE INHIBITORS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP;

CLOSTRIDIUM HISTOLYTICUM;

EID: 0037320183     PISSN: 14756366     EISSN: None     Source Type: Journal    
DOI: 10.1080/1475636021000049735     Document Type: Article

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