Serotonin type-4 (5-HT4) receptors as therapeutic targets: 5-HT4 receptor antagonists

Current Medicinal Chemistry - Central Nervous System Agents

Volumn 3, Issue 1, 2003, Pages 37-42

  Mattes, Henri ^a   Pfannkuche, Hans Juergen ^a  

^a NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

1 METHYL 3 INDOLECARBOXYLIC ACID [1 [2 (METHYLSULFONYLAMINO)ETHYL] 4 PIPERIDINYLMETHYL] ESTER; 2,3 DIHYDRO 2 OXO 1 BENZIMIDAZOLECARBOXYLIC ACID 6 METHOXY 3ALPHA TROPANYL ESTER; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 2 (DIETHYLAMINO)ETHYL ESTER; 4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 3 PIPERIDINOPROPYL ESTER; 5 FLUORO 2 METHOXY 1H INDOLE 3 CARBOXYLIC ACID 1 [2 (METHYLSULFONAMIDO)ETHYL] 4 PIPERIDINYLMETHYL ESTER; 6 CHLORO N [(HEXAHYDRO 1H PYRROLIZIN 1 YL)METHYL]IMIDAZO[1,2 A]PYRIDINE 8 CARBOXAMIDE; 8 AMINO 7 CHLORO 1,4 BENZODIOXAN 5 CARBOXYLIC ACID 1 BUTYL 4 PIPERIDINYLMETHYL ESTER; N [2 [4 (1 ADAMANTANECARBOXAMIDO) 1 PIPERIDINYL]ETHYL] 1 ISOPROPYL 1H INDAZOLE 3 CARBOXAMIDE; PIBOSEROD; RS 39604; SDZ 219048; SEROTONIN 4 ANTAGONIST; SEROTONIN 4 RECEPTOR; TROPISETRON; UNCLASSIFIED DRUG;

CARDIOVASCULAR DISEASE; CLINICAL TRIAL; COMPETITIVE INHIBITION; DIARRHEA; DRUG ACTIVITY; DRUG INDICATION; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG TARGETING; GASTROINTESTINAL DISEASE; HEART ATRIUM ARRHYTHMIA; HEART ATRIUM FIBRILLATION; HUMAN; INTESTINE MOTILITY; IRRITABLE COLON; NEUROLOGIC DISEASE; NONHUMAN; PHARMACOLOGICAL BLOCKING; PROPHYLAXIS; RECEPTOR BLOCKING; REVIEW;

EID: 0037284426     PISSN: 15680150     EISSN: None     Source Type: Journal    
DOI: 10.2174/1568015033357742     Document Type: Review

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