LY353433, a potent, orally effective, long-acting 5-HT4 receptor antagonist: Comparison to cisapride and RS23597-190

Journal of Pharmacology and Experimental Therapeutics

Volumn 277, Issue 1, 1996, Pages 97-104

  Cohen, Marlene L ^a   Bloomquist, William ^a   Schaus, John M ^a   Thompson, Dennis C ^a   Susemichel, Alice D ^a   Calligaro, David O ^a   Cohen, Ilene ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINO 5 CHLORO 2 METHOXYBENZOIC ACID 3 PIPERIDINOPROPYL ESTER; 8 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 5 PHENYL 1H 3 BENZAZEPIN 7 OL HYDROGEN MALEATE; CARBACHOL; CISAPRIDE; FLUNITRAZEPAM; KETANSERIN; MEPYRAMINE; MUSCIMOL; N [2 [4 (1 ADAMANTANECARBOXAMIDO) 1 PIPERIDINYL]ETHYL] 1 ISOPROPYL 1H INDAZOLE 3 CARBOXAMIDE; PRAZOSIN; RACLOPRIDE; RAUWOLSCINE; SEROTONIN ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DOSE RESPONSE; DOSE TIME EFFECT RELATION; DRUG ABSORPTION; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SAFETY; ESOPHAGUS FUNCTION; FEMALE; INTRAVENOUS DRUG ADMINISTRATION; NONHUMAN; ORAL DRUG ADMINISTRATION; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR BLOCKING;

ADAMANTANE; ADMINISTRATION, ORAL; AMINOBENZOIC ACIDS; ANIMALS; CISAPRIDE; ESOPHAGUS; FEMALE; INDAZOLES; MALE; MUSCLE RELAXATION; PIPERIDINES; RATS; RATS, INBRED F344; RATS, SPRAGUE-DAWLEY; RATS, WISTAR; SEROTONIN ANTAGONISTS;

EID: 0030431051     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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