Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs): Discovery of capromorelin

Bioorganic and Medicinal Chemistry

Volumn 11, Issue 4, 2003, Pages 581-590

  Carpino, Philip A ^a   Lefker, Bruce A ^a   Toler, Steven M ^a   Pan, Lydia C ^a   Hadcock, John R ^a   Cook, Ewell R ^a   DiBrino, Joseph N ^a   Campeta, Anthony M ^a   DeNinno, Shari L ^a   Chidsey Frink, Kristin L ^a   Hada, William A ^a   Inthavongsay, John ^a   Mangano, F Michael ^a   Mullins, Michelle A ^a   Nickerson, David F ^a   Ng, Oicheng ^a   Pirie, Christine M ^a   Ragan, John A ^a   Rose, Colin R ^a   Tess, David A ^a   Wright, Ann S ^a   Yu, Li ^a   Zawistoski, Michael P ^a   DaSilva Jardine, Paul A ^a   Wilson, Theresa C ^a   Thompson, David D ^a   more..

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CAPROMORELIN; DIPEPTIDE DERIVATIVE; GHRELIN; GROWTH HORMONE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG POTENCY; DRUG SYNTHESIS; FEMALE; GROWTH HORMONE BLOOD LEVEL; HUMAN; HUMAN CELL; INTESTINE ABSORPTION; NONHUMAN; RAT;

ANIMALS; CELLS, CULTURED; CHEMISTRY, PHYSICAL; DIPEPTIDES; DNA, COMPLEMENTARY; DOGS; DRUG DESIGN; FEMALE; GROWTH HORMONE; HALF-LIFE; HUMANS; INDICATORS AND REAGENTS; INDOLES; MAGNETIC RESONANCE SPECTROSCOPY; PIPERIDINES; PITUITARY GLAND; PYRAZOLES; RATS; RATS, SPRAGUE-DAWLEY; RATS, WISTAR; SOLUBILITY; SPIRO COMPOUNDS;

ANIMALIA; CANIS FAMILIARIS; RODENTIA;

EID: 0037249113     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00433-9     Document Type: Article

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