Unique insecticide specificity of human homomeric ρ1 GABAC receptor

Toxicology Letters

Volumn 129, Issue 1-2, 2002, Pages 47-53

  Ratra, Gurpreet S ^a   Erkkila, Brian E ^b   Weiss, David S ^b   Casida, John E ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b University of Alabama at Birmingham   (United States)

Author keywords

Aminobutyric acid; 3H EBOB; Binding site specificity; GABA induced currents; GABAC 1 receptor; Insecticide

Indexed keywords

4 AMINOBUTYRIC ACID C RECEPTOR; 4 PROPYL 4' ETHYNYLBICYCLOORTHOBENZOATE; 4' CYANO 4 SEC BUTYLBICYCLOORTHOBENZOATE; BENZOIC ACID DERIVATIVE; ENDOSULFAN; FIPRONIL; INSECTICIDE; PICROTOXIN; TERT BUTYLBICYCLOPHOSPHOROTHIOATE; TRITIUM; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; COMPETITIVE INHIBITION; CONTROLLED STUDY; EMBRYO; HUMAN; HUMAN CELL; NONHUMAN; OOCYTE; PRIORITY JOURNAL; PROTEIN EXPRESSION; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR SENSITIVITY; XENOPUS;

BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING SITES; CHLORIDE CHANNELS; GAMMA-AMINOBUTYRIC ACID; HUMANS; INSECTICIDES; MEMBRANE POTENTIALS; RECEPTORS, GABA; RECEPTORS, GABA-A; SENSITIVITY AND SPECIFICITY;

EID: 0037165506     PISSN: 03784274     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-4274(01)00471-4     Document Type: Article

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