GABA receptor subunit composition relative to insecticide potency and selectivity

Toxicology Letters

Volumn 122, Issue 3, 2001, Pages 215-222

  Ratra, Gurpreet S ^a   Casida, John E ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Endosulfan; Aminobutryic acid; 3H EBOB; Binding site specificity; Fipronil; GABA receptor; GABA receptor subunits; Insecticide; Lindane; Subunit composition

Indexed keywords

4 AMINOBUTYRIC ACID ALPHA1 RECEPTOR; 4 AMINOBUTYRIC ACID ALPHA6 RECEPTOR; 4 AMINOBUTYRIC ACID BETA1 RECEPTOR; 4 AMINOBUTYRIC ACID BETA3 RECEPTOR; 4 AMINOBUTYRIC ACID GAMMA2 RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR; 4 PROPYL 4' ETHYNYLBICYCLOORTHOBENZOATE; BENZOIC ACID DERIVATIVE; ENDOSULFAN; FIPRONIL; INSECTICIDE; LINDANE; RECEPTOR SUBUNIT; RECOMBINANT RECEPTOR; TRITIUM; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BINDING SITE; BRAIN; CHEMICAL STRUCTURE; CONTROLLED STUDY; CORRELATION FUNCTION; DATA ANALYSIS; HOUSE FLY; HUMAN; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RECEPTOR BINDING; RECEPTOR SENSITIVITY; REGULATORY MECHANISM; SEQUENCE HOMOLOGY; STRUCTURE ACTIVITY RELATION;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING SITES; BINDING, COMPETITIVE; BRAIN; DIPTERA; ENDOSULFAN; HUMANS; INSECTICIDES; LINDANE; PROTEIN CONFORMATION; PYRAZOLES; RECEPTORS, GABA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035816185     PISSN: 03784274     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0378-4274(01)00366-6     Document Type: Article

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