Parallel synthesis and anti-malarial activity of a sulfonamide library

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 18, 2002, Pages 2595-2598

  Ryckebusch, A ^a   Deprez Poulain R ^a   Debreu Fontaine, M A ^a   Vandaele, R ^a   Mouray, E ^b   Grellier, P ^b   Sergheraert, C ^a  

^a CNRS   (France)

^b MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIMALARIAL AGENT; CHLOROQUINE; SULFONAMIDE;

ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SYNTHESIS; FLUORESCENCE; HUMAN; HUMAN CELL; NONHUMAN; PLASMODIUM FALCIPARUM;

ANTIMALARIALS; CELL LINE; HUMANS; MICROSCOPY, FLUORESCENCE; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

PLASMODIUM FALCIPARUM;

EID: 0037119799     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00475-4     Document Type: Article

References (14)

1. Van Est H.G., Skamene G.E., Schurr E. Clin. Invest. Med. 16:1993;285.
2. White N.J. J. Antimicrob. Chemother. 30:1992;571.
3. WHO, 1999. Report of Infectious Diseases; World Health Organization: Geneva.
4. Dorn A., Stoffel R., Matile H., Bubendorf A., Ridley R.G. Nature. 374:1995;269.
5. Dorn A., Vippagunta S.R., Matile H., Jaquet C., Vennerstrom J.L., Ridley R.G. Biochem. Pharmacol. 55:1998;727.
6. Krogstad D.J., Gluzman I.Y., Kyle D.E., Oduola A.M., Martin S.K., Milhous W.K., Schlesinger P.H. Science. 238:1987;1283.
7. Reed M.B., Saliba K.J., Caruana S.R., Kirk K., Cowman A.F. Nature. 403:2000;906.
8. Vennerstrom J.L., Ellis W.Y., Ager A.L., Andersen S.L., Gerena L., Milhous W.K. J. Med. Chem. 35:1992;2129.
9. Raynes K., Galatis D., Cowman A.F., Tilley L., Deady L.W. J. Med. Chem. 38:1995;204.
10. Girault S., Grellier P., Berecibar A., Maes L., Mouray E., Lemière P., Debreu M.A., Davioud-Charvet E., Sergheraert C. J. Med. Chem. 43:2000;2646.
11. Unpublished results.
12. Desjardins R.E., Canfield C.J., Haynes J.D., Chulay J.D. Antimicrob. Agents. Chemother. 16:1979;710.
13. Delarue S., Girault S., Maes L., Debreu-Fontaine M.-A., Labaïed M., Grelleir P., Sergheraert C. J. Med. Chem. 44:2001;2827.
14. Experiments on log D in progress.