Phosphorylation of Ser360 in the third intracellular loop of the α2A-adrenoceptor during protein kinase C-mediated desensitization

European Journal of Pharmacology

Volumn 437, Issue 1-2, 2002, Pages 41-46

  Liang, Mei ^a   Eason, Margaret G ^a   Theiss, Cheryl T ^a   Liggett, Stephen B ^a  

^a UNIVERSITY OF CINCINNATI COLLEGE OF MEDICINE   (United States)

Author keywords

Desensitization; Mutation; Phosphorylation; Protein kinase C

Indexed keywords

ALPHA 2A ADRENERGIC RECEPTOR; BRIMONIDINE; CALCIUM; INOSITOL PHOSPHATE; PHORBOL 13 ACETATE 12 MYRISTATE; PROTEIN KINASE C; SERINE; ALPHA 2 ADRENERGIC RECEPTOR; INOSITOL 1,4,5 TRISPHOSPHATE; RECEPTOR, ADRENERGIC, ALPHA 2A; RECEPTOR, ADRENERGIC, ALPHA-2A;

AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; CALCIUM CELL LEVEL; CALCIUM TRANSPORT; CONTROLLED STUDY; DESENSITIZATION; ENZYME ACTIVATION; LIGAND BINDING; MUTATION; NONHUMAN; PHOSPHORYLATION; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; REGULATORY MECHANISM; SIGNAL TRANSDUCTION; ANIMAL; BINDING COMPETITION; BINDING SITE; CHO CELL; DRUG EFFECT; GENETICS; GENOTYPE; HAMSTER; HUMAN; METABOLISM; RADIOASSAY;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CALCIUM; CHO CELLS; CRICETINAE; GENOTYPE; HUMANS; INOSITOL 1,4,5-TRISPHOSPHATE; MUTATION; PHOSPHORYLATION; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA-2; SERINE; TETRADECANOYLPHORBOL ACETATE;

EID: 0037082359     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(02)01280-3     Document Type: Article

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