-
1
-
-
33748237769
-
-
(a) Früchtel, J. S.; Jung, G. Angew. Chem., Int. Ed. Engl. 1996, 35, 17.
-
(1996)
Angew. Chem., Int. Ed. Engl.
, vol.35
, pp. 17
-
-
Früchtel, J.S.1
Jung, G.2
-
3
-
-
0029074627
-
-
Han, H.; Wolfe, M. M.; Brenner, S.; Janda, K. D. Proc. Natl. Acad. Sci. U.S.A. 1995, 92, 6419.
-
(1995)
Proc. Natl. Acad. Sci. U.S.A.
, vol.92
, pp. 6419
-
-
Han, H.1
Wolfe, M.M.2
Brenner, S.3
Janda, K.D.4
-
6
-
-
0031098534
-
-
Reviews on liquid-phase organic synthesis (LPOS): (a) Gravert, D. J.; Janda, K. D. Chem. Rev. 1997, 97, 489. (b) Harwig, C. W.; Gravert, D. J.; Janda, K. D. Chemtracts: Org. Chem. 1999, 12, 1. (c) Gravert, D. J.; Janda, K. D. In Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series; Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC, 1996, 118-127. (d) Vandersteen, A. M.; Han, H.; Janda, K. D. Mol. Diversity 1996, 2, 89. (e) For a recent example of LPOS, see: Annunziata, R; Benaglia, M.; Cinquini, M.; Cozzi, F. Chem.-Eur. J. 2000, 6, 133.
-
(1997)
Chem. Rev.
, vol.97
, pp. 489
-
-
Gravert, D.J.1
Janda, K.D.2
-
7
-
-
0032848810
-
-
Reviews on liquid-phase organic synthesis (LPOS): (a) Gravert, D. J.; Janda, K. D. Chem. Rev. 1997, 97, 489. (b) Harwig, C. W.; Gravert, D. J.; Janda, K. D. Chemtracts: Org. Chem. 1999, 12, 1. (c) Gravert, D. J.; Janda, K. D. In Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series; Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC, 1996, 118-127. (d) Vandersteen, A. M.; Han, H.; Janda, K. D. Mol. Diversity 1996, 2, 89. (e) For a recent example of LPOS, see: Annunziata, R; Benaglia, M.; Cinquini, M.; Cozzi, F. Chem.-Eur. J. 2000, 6, 133.
-
(1999)
Chemtracts: Org. Chem.
, vol.12
, pp. 1
-
-
Harwig, C.W.1
Gravert, D.J.2
Janda, K.D.3
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8
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3142538092
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Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC
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Reviews on liquid-phase organic synthesis (LPOS): (a) Gravert, D. J.; Janda, K. D. Chem. Rev. 1997, 97, 489. (b) Harwig, C. W.; Gravert, D. J.; Janda, K. D. Chemtracts: Org. Chem. 1999, 12, 1. (c) Gravert, D. J.; Janda, K. D. In Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series; Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC, 1996, 118-127. (d) Vandersteen, A. M.; Han, H.; Janda, K. D. Mol. Diversity 1996, 2, 89. (e) For a recent example of LPOS, see: Annunziata, R; Benaglia, M.; Cinquini, M.; Cozzi, F. Chem.-Eur. J. 2000, 6, 133.
-
(1996)
Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series
, pp. 118-127
-
-
Gravert, D.J.1
Janda, K.D.2
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9
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0030252431
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Reviews on liquid-phase organic synthesis (LPOS): (a) Gravert, D. J.; Janda, K. D. Chem. Rev. 1997, 97, 489. (b) Harwig, C. W.; Gravert, D. J.; Janda, K. D. Chemtracts: Org. Chem. 1999, 12, 1. (c) Gravert, D. J.; Janda, K. D. In Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series; Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC, 1996, 118-127. (d) Vandersteen, A. M.; Han, H.; Janda, K. D. Mol. Diversity 1996, 2, 89. (e) For a recent example of LPOS, see: Annunziata, R; Benaglia, M.; Cinquini, M.; Cozzi, F. Chem.-Eur. J. 2000, 6, 133.
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(1996)
Mol. Diversity
, vol.2
, pp. 89
-
-
Vandersteen, A.M.1
Han, H.2
Janda, K.D.3
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10
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0033985668
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Reviews on liquid-phase organic synthesis (LPOS): (a) Gravert, D. J.; Janda, K. D. Chem. Rev. 1997, 97, 489. (b) Harwig, C. W.; Gravert, D. J.; Janda, K. D. Chemtracts: Org. Chem. 1999, 12, 1. (c) Gravert, D. J.; Janda, K. D. In Molecular Diversity and Combinatorial Synthesis: Libraries and Drug Discovery, ACS Symposium Series; Chaiken, I. M.; Janda, K. D., Eds.; American Chemical Society: Washington DC, 1996, 118-127. (d) Vandersteen, A. M.; Han, H.; Janda, K. D. Mol. Diversity 1996, 2, 89. (e) For a recent example of LPOS, see: Annunziata, R; Benaglia, M.; Cinquini, M.; Cozzi, F. Chem.-Eur. J. 2000, 6, 133.
-
(2000)
Chem.-Eur. J.
, vol.6
, pp. 133
-
-
Annunziata, R.1
Benaglia, M.2
Cinquini, M.3
Cozzi, F.4
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11
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0030883333
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2 at -78 °C. To circumvent this problem Janda et al. have successfully used noncross-linked chloromethylated polystyrene (NCPS) as a soluble polymer support: Chen, S.; Janda, K. D. J. Am. Chem. Soc. 1997, 119, 8724.
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(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 8724
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Chen, S.1
Janda, K.D.2
-
12
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0032511939
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Zhao, X. Y.; Metz, W. A.; Sieber, F.; Janda, K. D. Tetrahedron Lett. 1998, 39, 8433.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 8433
-
-
Zhao, X.Y.1
Metz, W.A.2
Sieber, F.3
Janda, K.D.4
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15
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0345764879
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note
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A search in MDDR (MDL data base) revealed the presence of more than 250 structures based on the isoxazole scaffold and endowed with several pharmacological activities used for analgesia, inflammation, immunology and CNS diseases (such as anxiety, memory impairment, depression, Parkinson's and stroke).
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16
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0032563904
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The first example of a liquid-phase 1,3-dipolar cycloaddition reaction was reported by Norris et al.: Moore, M.; Norris, P. Tetrahedron Lett. 1998, 39, 7027.
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(1998)
Tetrahedron Lett.
, vol.39
, pp. 7027
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Moore, M.1
Norris, P.2
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17
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0032560063
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(a) Shankar, B. B.; Yang, D. Y.; Girton, S.; Ganguly, A. K. Tetrahedron Lett. 1998, 39, 2447.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 2447
-
-
Shankar, B.B.1
Yang, D.Y.2
Girton, S.3
Ganguly, A.K.4
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18
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0034729961
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(b) Batra, S.; Rastogi, S. K.; Kundu, B.; Patra, A.; Bhaduri, A. P. Tetrahedron Lett. 2000, 41, 5971.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 5971
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Batra, S.1
Rastogi, S.K.2
Kundu, B.3
Patra, A.4
Bhaduri, A.P.5
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19
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0035812802
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Luca, L. D.; Giacomelli, G.; Riu, A. J. Org. Chem. 2001, 66, 6823.
-
(2001)
J. Org. Chem.
, vol.66
, pp. 6823
-
-
Luca, L.D.1
Giacomelli, G.2
Riu, A.3
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