2D-QSAR in hydroxamic acid derivatives as peptide deformylase inhibitors and antibacterial agents

Bioorganic and Medicinal Chemistry

Volumn 10, Issue 12, 2002, Pages 3713-3716

  Gupta, Manish K ^a,b   Mishra, Pradeep ^a,b   Prathipati, Philip ^a   Saxena, Anil K ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

^b DR H S GOUR UNIVERSITY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; ENZYME INHIBITOR; FERROUS ION; HYDROXAMIC ACID DERIVATIVE; MATRIX METALLOPROTEINASE; PEPTIDE DEFORMYLASE; PROTEINASE;

ANTIBACTERIAL ACTIVITY; ARTICLE; BINDING SITE; CELL FREE SYSTEM; CONTROLLED STUDY; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME ISOLATION; ESCHERICHIA COLI; HYDROPHOBICITY; MORAXELLA CATARRHALIS; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION;

AMIDOHYDROLASES; AMINOPEPTIDASES; ANTI-BACTERIAL AGENTS; BACTERIAL PROTEINS; BINDING SITES; ESCHERICHIA COLI; HYDROPHOBICITY; HYDROXAMIC ACIDS; MORAXELLA (BRANHAMELLA) CATARRHALIS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; STRUCTURE-ACTIVITY RELATIONSHIP;

BACTERIA (MICROORGANISMS); ESCHERICHIA COLI; MORAXELLA CATARRHALIS;

EID: 0036979118     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00421-2     Document Type: Article

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