메뉴 건너뛰기




Volumn 96, Issue 6, 2002, Pages 677-683

The effect of 10α-trifluoromethylhydroartemisinin on Plasmodium berghei infection and its toxicity in experimental animals

Author keywords

10 trifluoromethylhydroartemisinin; Artemisinin; Chemotherapy; Dihydroartemisin; Malaria; Plasmodium berghei

Indexed keywords

ARTEMISININ DERIVATIVE; CHLOROQUINE; DIHYDROARTEMISININ;

EID: 0036880638     PISSN: 00359203     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0035-9203(02)90350-0     Document Type: Article
Times cited : (17)

References (31)
  • 4
    • 0028271047 scopus 로고
    • In-vitro reversal of chloroquine resistance with chlorpheniramine against African isolates of Plasmodium falciparum
    • Basco, L. K. & Le Bras, J. (1994). In-vitro reversal of chloroquine resistance with chlorpheniramine against African isolates of Plasmodium falciparum. Japanese Journal of Medical Science and Biology, 47, 59-63.
    • (1994) Japanese Journal of Medical Science and Biology , vol.47 , pp. 59-63
    • Basco, L.K.1    Le Bras, J.2
  • 5
    • 0004071134 scopus 로고
    • Molécules antipaludiques
    • Paris: Masson Publishers
    • Basco, L. K., Ruggeri, C. & Le Bras, J. (1994). Molécules antipaludiques. Me'anisme de résistance, volume 2. Paris: Masson Publishers, pp. 74-75.
    • (1994) Me'anisme De Résistance , vol.2 , pp. 74-75
    • Basco, L.K.1    Ruggeri, C.2    Le Bras, J.3
  • 6
    • 0025963466 scopus 로고
    • Preparation of trifluoromethyl ketones and related fluorinated ketones
    • Bégué, J. P. & Bonnet-Delpon, D. (1991). Preparation of trifluoromethyl ketones and related fluorinated ketones. Tetrahedron, 47, 3207-3254.
    • (1991) Tetrahedron , vol.47 , pp. 3207-3254
    • Bégué, J.P.1    Bonnet-Delpon, D.2
  • 8
    • 0344639143 scopus 로고
    • Detection of a system of microsomal monooxygenases in a malaria parasite of rodents, Plasmodium berghei
    • Chekhonadskikh, T. V., Polyakova, N. E., Pankova, T. G. & Salganik, R. I. (1987). Detection of a system of microsomal monooxygenases in a malaria parasite of rodents, Plasmodium berghei. Biochemistry-Moscow, 52, 327-331.
    • (1987) Biochemistry-Moscow , vol.52 , pp. 327-331
    • Chekhonadskikh, T.V.1    Polyakova, N.E.2    Pankova, T.G.3    Salganik, R.I.4
  • 9
    • 0026239217 scopus 로고
    • Identification of the in vivo metabolites of the antimalarial arteether by thermospray high performance liquid chromatography/mass spectrometry
    • Chi, H. T., Ramu, K., Barker, J. K., Hufford, C. D., Lee, I. S., Zeng, Y. L. & McChesney, J. D. (1991). Identification of the in vivo metabolites of the antimalarial arteether by thermospray high performance liquid chromatography/mass spectrometry. Biological Mass Spectrometry, 20, 609-628.
    • (1991) Biological Mass Spectrometry , vol.20 , pp. 609-628
    • Chi, H.T.1    Ramu, K.2    Barker, J.K.3    Hufford, C.D.4    Lee, I.S.5    Zeng, Y.L.6    McChesney, J.D.7
  • 10
    • 0020097276 scopus 로고
    • Studies on the toxicity of quinghaosu and its derivatives
    • China Cooperative Research Group on Qinghaosu and its Derivatives as Antimalarials
    • China Cooperative Research Group on Qinghaosu and its Derivatives as Antimalarials (1982a). Studies on the toxicity of quinghaosu and its derivatives. Journal of Traditional Chinese Medicine, 2, 31-38.
    • (1982) Journal of Traditional Chinese Medicine , vol.2 , pp. 31-38
  • 11
    • 0020097272 scopus 로고
    • Clinical studies on the treatment of malaria with quinghaosu and its derivatives
    • China Cooperative Research Group on Qinghaosu and its Derivatives as Antimalarials
    • China Cooperative Research Group on Qinghaosu and its Derivatives as Antimalarials (1982b). Clinical studies on the treatment of malaria with quinghaosu and its derivatives. Journal of Traditional Chinese Medicine, 2, 45-50.
    • (1982) Journal of Traditional Chinese Medicine , vol.2 , pp. 45-50
  • 12
    • 0019174245 scopus 로고
    • Activities of 25 derivatives of artemisinine against chloroquine-resistant Plasmodium berghei
    • Gu, H. M., Lu, B. F. & Qu, Z. X. (1980). Activities of 25 derivatives of artemisinine against chloroquine-resistant Plasmodium berghei. Acta Pharmacological Sinica, 1, 48-50.
    • (1980) Acta Pharmacological Sinica , vol.1 , pp. 48-50
    • Gu, H.M.1    Lu, B.F.2    Qu, Z.X.3
  • 13
    • 85031227378 scopus 로고    scopus 로고
    • Study on the toxicology of natri artesunate and its effect to the other drugs metabolism in experimental animals
    • PhD thesis, Hanoi Medical University, Viet Nam
    • Huong, N. T. G. (1997). Study on the toxicology of natri artesunate and its effect to the other drugs metabolism in experimental animals. PhD thesis, Hanoi Medical University, Viet Nam.
    • (1997)
    • Huong, N.T.G.1
  • 14
    • 0028068979 scopus 로고
    • Comparison of in vivo and in vitro antimalarial activity of artemisinin, dihydroartemisinin and sodium artesunate in the Plasmodium berghei-rodent model
    • Janse, C. J., Waters, A. P., Kos, J. & Lugt, C. B. (1994). Comparison of in vivo and in vitro antimalarial activity of artemisinin, dihydroartemisinin and sodium artesunate in the Plasmodium berghei-rodent model. International Journal for Parasitology, 24, 589-594.
    • (1994) International Journal for Parasitology , vol.24 , pp. 589-594
    • Janse, C.J.1    Waters, A.P.2    Kos, J.3    Lugt, C.B.4
  • 16
    • 0021948029 scopus 로고
    • Qinghaosu (artemisinin): An antimalarial drug from China
    • Klayman, D. L. (1985). Qinghaosu (artemisinin): an antimalarial drug from China. Science, 288, 1049-1055.
    • (1985) Science , vol.288 , pp. 1049-1055
    • Klayman, D.L.1
  • 18
    • 0028951562 scopus 로고
    • Antimalarial activity of new dihydroartemisinin derivatives. 6. α-Alkylbenzylic ethers
    • Lin, A. J. & Miller, R. E. (1995). Antimalarial activity of new dihydroartemisinin derivatives. 6. α-Alkylbenzylic ethers. Journal of Medicinal Chemistry, 38, 764-770.
    • (1995) Journal of Medicinal Chemistry , vol.38 , pp. 764-770
    • Lin, A.J.1    Miller, R.E.2
  • 19
    • 0030963326 scopus 로고    scopus 로고
    • Antimalarial activity of new hydro artemisinin derivatives. 7.4-(p-substituted phenyl)- 4 (R or S)- [10(α or β) dihydroartemisinin oxy] butyric acids
    • Lin, A. J., Zikry, A. B. & Kyle. D. E. (1997). Antimalarial activity of new hydro artemisinin derivatives. 7.4-(p-substituted phenyl)- 4 (R or S)- [10(α or β) dihydroartemisinin oxy] butyric acids. Journal of Medicinal Chemistry, 40, 1396-1400.
    • (1997) Journal of Medicinal Chemistry , vol.40 , pp. 1396-1400
    • Lin, A.J.1    Zikry, A.B.2    Kyle, D.E.3
  • 20
    • 0023110445 scopus 로고
    • The chemistry, pharmacology, and clinical applications of qinghaosu (artemisinin) and its derivatives
    • Luo, X. D. & Shen, C. C. (1987). The chemistry, pharmacology, and clinical applications of qinghaosu (artemisinin) and its derivatives. Medicinal Research Review, 7, 29-52.
    • (1987) Medicinal Research Review , vol.7 , pp. 29-52
    • Luo, X.D.1    Shen, C.C.2
  • 22
    • 0344207602 scopus 로고
    • Techniques of drug evaluation I: Primary screening
    • Peters, W. (editor). London: Academic Press
    • Peters, W. (1987). Techniques of drug evaluation I: primary screening. In: Chemotherapy and Drug Resistance in Malaria, volume 1, Peters, W. (editor). London: Academic Press, pp. 100-123.
    • (1987) Chemotherapy and Drug Resistance in Malaria , vol.1 , pp. 100-123
    • Peters, W.1
  • 23
    • 0028788118 scopus 로고
    • Synthesis and antimalarial activities of several fluorinated artemisinin derivatives
    • Pu, Y. M., Torok, D. S., Ziffer, H., Pan, X. Q. & Meshnick, S. R. (1995). Synthesis and antimalarial activities of several fluorinated artemisinin derivatives. Journal of Medicinal Chemistry, 38, 4120-4124.
    • (1995) Journal of Medicinal Chemistry , vol.38 , pp. 4120-4124
    • Pu, Y.M.1    Torok, D.S.2    Ziffer, H.3    Pan, X.Q.4    Meshnick, S.R.5
  • 24
    • 0029071407 scopus 로고
    • Synthesis, characterization, and antimalarial activity of the glucuronides of the hydroxylated metabolites of arteether
    • Ramu, K. & Baker, J. K. (1995). Synthesis, characterization, and antimalarial activity of the glucuronides of the hydroxylated metabolites of arteether. Journal of Medicinal Chemistry, 38, 1911-1921.
    • (1995) Journal of Medicinal Chemistry , vol.38 , pp. 1911-1921
    • Ramu, K.1    Baker, J.K.2
  • 25
    • 0024851248 scopus 로고
    • Studies of qinghaosu and its active derivatives in biological materials and their pharmacokineties
    • Peking Union Medical College
    • Song, Z. Y. & Zhao, K. C. (1989). Studies of qinghaosu and its active derivatives in biological materials and their pharmacokineties. Proceedings of the Chinese Academy of Medicinal Science, Peking Union Medical College, 4, 229-234.
    • (1989) Proceedings of the Chinese Academy of Medicinal Science , vol.4 , pp. 229-234
    • Song, Z.Y.1    Zhao, K.C.2
  • 28
    • 85031213208 scopus 로고    scopus 로고
    • Estimate the effect of dihydroartemisinin (the produce of Vietnam) in mice infected with a P. berghei experimental model
    • Hanoi: National Institute of Malariology, Parasitology and Entomology, internal document, no. 4
    • Tien, N. T., Lien, L. K., Cong, L. D. Nhan, D. H., Huong, N. M., Hanh, N. T., Xuan, D. T., Tao, N. D. & Ha, N. T. H. (2000). Estimate the effect of dihydroartemisinin (the produce of Vietnam) in mice infected with a P. berghei experimental model. In: Information on Malaria Prevention and Parasite Diseases. Hanoi: National Institute of Malariology, Parasitology and Entomology, internal document, no. 4, pp. 26-32.
    • (2000) Information on Malaria Prevention and Parasite Diseases , pp. 26-32
    • Tien, N.T.1    Lien, L.K.2    Cong, L.D.3    Nhan, D.H.4    Huong, N.M.5    Hanh, N.T.6    Xuan, D.T.7    Tao, N.D.8    Ha, N.T.H.9
  • 30
    • 0000955998 scopus 로고
    • Study on the chemistry of qinghaosu (artemisinin)
    • Wu, Y. L. & Li, Y. (1995). Study on the chemistry of qinghaosu (artemisinin). Medicinal Chemistry Review, 5, 569-586.
    • (1995) Medicinal Chemistry Review , vol.5 , pp. 569-586
    • Wu, Y.L.1    Li, Y.2
  • 31
    • 0022219529 scopus 로고
    • Studies on systemic pharmacological effects of artesunate
    • Yi Zhao (1985). Studies on systemic pharmacological effects of artesunate. Journal of Tropical Medicine and Hygiene, 88, 391-396.
    • (1985) Journal of Tropical Medicine and Hygiene , vol.88 , pp. 391-396
    • Zhao, Y.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.