Synthesis and β1-, β2-adrenergic receptor binding studies of 4-acylamino-substituted phenoxypropanolamine and 5-acylamino-substituted naphthyloxypropanolamine derivatives

Arzneimittel-Forschung/Drug Research

Volumn 52, Issue 9, 2002, Pages 654-663

  Jindal, Dharam Paul ^a   Coumar, Mohane S ^a   Bruni, Giancarlo ^a   Massarelli, Paola ^a  

^a PANJAB UNIVERSITY   (India)

Author keywords

Aryloxypropanolamines, 1 and 2 adrenergic receptor binding affinity; CAS 318 98 9; Dihydroalprenolol, radiolabelled; Propranolol; Adrenergic blocking agents

Indexed keywords

3 ISOPROPYLAMINO 1 (7 METHYL 4 INDANYLOXY) 2 BUTANOL; BETA 1 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; N [5 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY)NAPHTHALEN 1 YL]ACETAMIDE; NAPHTHYLOXYPROPANOLAMINE DERIVATIVE; PHENOXYPROPANOLAMINE DERIVATIVE; PROPANOLAMINE DERIVATIVE; PROPRANOLOL; UNCLASSIFIED DRUG;

ADRENERGIC SYSTEM; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; ERYTHROCYTE MEMBRANE; LUNG; MALE; NONHUMAN; RAT; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; TURKEY (BIRD);

EID: 0036380852     PISSN: 00044172     EISSN: None     Source Type: Journal    
DOI: 10.1055/s-0031-1299947     Document Type: Article

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