메뉴 건너뛰기




Volumn 301, Issue 2, 2002, Pages 661-671

Agonist, antagonist, and inverse agonist characteristics of TIPP (H-Tyr-Tic-Phe-Phe-OH), a selective δ-opioid receptor ligand

Author keywords

[No Author keywords available]

Indexed keywords

1,2,3,4 TETRAHYDROISOQUINOLINE PHENYLALANYLPHENYLALANINE; ADENYLATE CYCLASE; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; GUANINE NUCLEOTIDE; OPIATE AGONIST; OPIATE ANTAGONIST; SIGMA OPIATE RECEPTOR; SODIUM ION; UNCLASSIFIED DRUG;

EID: 0036228370     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.301.2.661     Document Type: Article
Times cited : (22)

References (37)
  • 4
    • 0002456732 scopus 로고
    • Transducin, rhodopsin and 3′5′-cyclic GMP phosphodiesterase: Typical G protein mediated transduction system
    • Iyengar R and Birnbaumer R, eds, Academic Press, San Diego
    • (1990) G Proteins , pp. 215-239
    • Chabre, M.1    Deterre, P.2
  • 5
    • 0015861774 scopus 로고
    • Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 percent inhibition (I50) of an enzymatic reaction
    • (1973) Biochem Pharmacol , vol.22 , pp. 3099-3108
    • Cheng, Y.1    Prusoff, W.H.2
  • 13
    • 0035083109 scopus 로고    scopus 로고
    • Inverse, protean, and ligand-selective agonism: Matters of receptor conformation
    • (2001) FASEB J , vol.15 , pp. 598-611
    • Kenakin, T.1
  • 15
    • 0020694935 scopus 로고
    • Opiate regulation of adenosine 3′:5′-cyclic monophosphate level in neuroblastoma X glioma NG108-15 hybrid cells. Relationship between receptor occupancy and effect
    • (1983) Mol Pharmacol , vol.23 , pp. 26-35
    • Law, P.Y.1    Hom, D.S.2    Loh, H.H.3
  • 16
    • 0020064965 scopus 로고
    • Comparison of opiate inhibition of adenylate cyclase activity in neuroblastoma N18tG2 and neuroblastoma x glioma NG108-15 hybrid cell lines
    • (1982) Mol Pharmacol , vol.21 , pp. 483-491
    • Law, P.Y.1    Koehler, J.E.2    Loh, H.H.3
  • 19
    • 0034955327 scopus 로고    scopus 로고
    • Chronic exposure to μ-opioid agonists produces constitutive activation of μ-opioid receptors in direct proportion to the efficacy of the agonist used for pretreatment
    • (2001) Mol Pharmacol , vol.60 , pp. 53-62
    • Liu, J.G.1    Prather, P.L.2
  • 35
    • 0031456986 scopus 로고    scopus 로고
    • Delta opioid modulation of the binding of guanosine-5′-O-(3- [35S]thio)triphosphate to NG-108-15 cell membranes: Characterization of agonist and inverse agonist effects
    • (1997) J Pharmacol Exp Ther , vol.283 , pp. 1276-1284
    • Szekeres, P.G.1    Traynor, J.R.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.