SCOPUS 정보 검색 플랫폼

Volumn 10, Issue 4, 2002, Pages 1009-1018

Guanidinium and aminoimidazolinium derivatives of N-(4-piperidyl)propanamides as potential ligands for μ opioid and I2-imidazoline receptors: Synthesis and pharmacological screening

(8) Montero, Ana a Goya, Pilar a Jagerovic, Nadine a Callado, Luis F b Meana, J Javier b Girón, Rocío c Goicoechea, Carlos c Martín, M Isabel c

a INSTITUTO DE QUÍMICA MÉDICA (Spain)

b UNIVERSITY OF THE BASQUE COUNTRY UPV EHU (Spain)

c UNIVERSIDAD REY JUAN CARLOS (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

ANALGESIC AGENT; ENKEPHALIN[2 DEXTRO ALANINE 4 METHYLPHENYLALANINE 5 GLYCINE]; ENKEPHALIN[2,5 DEXTRO PENICILLAMINE]; FENTANYL; GUANIDINE DERIVATIVE; IDAZOXAN; IMIDAZOLE DERIVATIVE; IMIDAZOLINE I2 RECEPTOR; MORPHINE; MU OPIATE RECEPTOR; N [1 (2 PHENETHYL) 4 PIPERIDYL] N (3 GUANIDINOPHENYL)PROPANAMIDE; N [1 (2 PHENETHYL) 4 PIPERIDYL] N (GUANIDINOPROPYL)PROPANAMIDE; N METHYL N [7 (1 PYRROLIDINYL) 1 OXASPIRO[4.5]DEC 8 YL]BENZENEACETAMIDE; NALOXONE; OPIATE RECEPTOR; RADIOLIGAND; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BRAIN; CELL MEMBRANE; CONTROLLED STUDY; DOSE RESPONSE; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; GUINEA PIG; HOT PLATE TEST; ILEUM; IN VITRO STUDY; MALE; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; STRUCTURE ACTIVITY RELATION; WRITHING TEST;

AMIDES; ANALGESICS; ANIMALS; DRUG EVALUATION, PRECLINICAL; GUANIDINE; GUINEA PIGS; IMIDAZOLES; LIGANDS; MALE; MICE; PIPERIDINES; RADIOLIGAND ASSAY; RECEPTORS, DRUG; RECEPTORS, OPIOID, MU; SENSATION; STRUCTURE-ACTIVITY RELATIONSHIP;

CAVIA PORCELLUS; SUS SCROFA;

EID: 0036170244 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00356-X Document Type: Article

Times cited : (29)

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