SB-334867-A antagonises orexin mediated excitation in the locus coeruleus

Neuropharmacology

Volumn 42, Issue 1, 2002, Pages 127-133

  Soffin, E M ^a   Evans, M L ^a   Gill, C H ^a   Harries, M H ^a   Benham, C D ^a   Davies, C H ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

Brain slices; Locus coeruleus; Orexin; Orexin receptors

Indexed keywords

1 (2 METHYLBENZOXAZOL 6 YL) 3 [1,5]NAPHTHYRIDIN 4 YLUREA; ALPHA ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; OREXIN A; OREXIN B; SB 334867 A; UNCLASSIFIED DRUG; UREA DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BRAIN NERVE CELL; CELL STRAIN; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG EFFECT; ELECTRON MICROSCOPY; LOCUS CERULEUS; MALE; NERVE CELL EXCITABILITY; NERVE CELL STIMULATION; NONHUMAN; NORADRENERGIC NERVE; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT;

ACTION POTENTIALS; ANIMALS; BENZOXAZOLES; CARRIER PROTEINS; ELECTROPHYSIOLOGY; INTRACELLULAR SIGNALING PEPTIDES AND PROTEINS; LOCUS COERULEUS; MALE; NEUROPEPTIDES; PATCH-CLAMP TECHNIQUES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, G-PROTEIN-COUPLED; RECEPTORS, METABOTROPIC GLUTAMATE; RECEPTORS, MUSCARINIC; RECEPTORS, NEUROPEPTIDE; UREA;

EID: 0036144494     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0028-3908(01)00156-3     Document Type: Article

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