Optimization of xanthones for antimalarial activity: The 3,6-bis-ω-diethylaminoalkoxyxanthone series

Antimicrobial Agents and Chemotherapy

Volumn 46, Issue 1, 2002, Pages 144-150

  Kelly, J X ^a   Winter, R ^a   Peyton, D H ^a   Hinrichs, D J ^a   Riscoe, M ^a  

^a PORTLAND VA MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3,6 BIS EPSILON (N,N DIETHYLAMINO)AMYLOXYXANTHONE; 3,6 BIS ZETA (N,N DIETHYLAMINO)HEXYLOXYXANTHONE; ANTIMALARIAL AGENT; CHLOROQUINE; HEME; HEMOZOIN; METALLOPORPHYRIN; PROPIONIC ACID; QUININE; UNCLASSIFIED DRUG; XANTHONE DERIVATIVE;

ANTIMALARIAL ACTIVITY; ARTICLE; BINDING AFFINITY; COMPLEX FORMATION; CONTROLLED STUDY; DRUG ACCUMULATION; DRUG POTENCY; HUMAN; HUMAN CELL; IC 50; MULTIDRUG RESISTANCE; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ALKANES; ANIMALS; ANTIMALARIALS; HEME; PARASITIC SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; STATISTICS; XANTHENES; XANTHONES;

EID: 0036135320     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/AAC.46.1.144-150.2002     Document Type: Article

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