A desensitization-selective potentiator of AMPA-type glutamate receptors

British Journal of Pharmacology

Volumn 136, Issue 7, 2002, Pages 1033-1041

  Sekiguchi, Masayuki ^a   Nishikawa, Kaori ^a   Aoki, Shunsuke ^a   Wada, Keiji ^a  

^a NATIONAL INSTITUTE OF NEUROSCIENCE   (Japan)

Author keywords

AMPA receptor; Deactivation; Desensitization; Flip; Flop; Kinetics; Model; PEPA; Simulation

Indexed keywords

4 [2 (PHENYLSULFONYLAMINO)ETHYLTHIO] 2,6 DIFLUOROPHENOXYACETAMIDE; ACETAMIDE; AMPA RECEPTOR; ANIRACETAM; CYCLOTHIAZIDE; GLUTAMATE RECEPTOR; UNCLASSIFIED DRUG; 2 PYRROLIDONE DERIVATIVE; 4 (2 (PHENYLSULFONYLAMINO)ETHYLTHIO) 2,6 DIFLUOROPHENOXYACETAMIDE; 4-(2-(PHENYLSULFONYLAMINO)ETHYLTHIO)-2,6-DIFLUOROPHENOXYACETAMIDE; BENZOTHIADIAZINE DERIVATIVE; GLUTAMATE RECEPTOR IONOTROPIC, AMPA 3; PHENOXYACETIC ACID DERIVATIVE;

ALLOSTERISM; ANIMAL CELL; ARTICLE; DESENSITIZATION; DRUG EFFECT; ENZYME ACTIVITY; HIPPOCAMPUS; LONG TERM POTENTIATION; NONHUMAN; PRIORITY JOURNAL; PYRAMIDAL NERVE CELL; RECEPTOR BINDING; RECEPTOR UPREGULATION; TASK PERFORMANCE; XENOPUS; ANIMAL; COMPARATIVE STUDY; IN VITRO STUDY; KINETICS; METABOLISM; OOCYTE; PATCH CLAMP; PHYSIOLOGY; RAT;

ALLOSTERIC REGULATION; ANIMAL; BENZOTHIADIAZINES; COMPARATIVE STUDY; IN VITRO; KINETICS; OOCYTES; PATCH-CLAMP TECHNIQUES; PHENOXYACETATES; PYRROLIDINONES; RATS; RECEPTORS, AMPA; SUPPORT, NON-U.S. GOV'T; XENOPUS; ANIMALS;

EID: 0036024238     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0704804     Document Type: Article

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