A novel allosteric potentiator of AMPA receptors: 4-[2- (phenylsulfonylamino)ethylthio]-2,6-difluoro-phenoxyacetamide

Journal of Neuroscience

Volumn 17, Issue 15, 1997, Pages 5760-5771

  Sekiguchi, Masayuki ^a   Fleck, Mark W ^b   Mayer, Mark L ^b   Takeo, Jiro ^c   Chiba, Yoshiyuki ^c   Yamashita, Shinya ^c   Wada, Keiji ^a  

^a NATIONAL INSTITUTE OF NEUROSCIENCE   (Japan)

^b EUNICE KENNEDY SHRIVER NATIONAL INSTITUTE OF CHILD HEALTH AND HUMAN DEVELOPMENT   (United States)

^c Central Research Laboratory   (Japan)

Author keywords

Allosteric modulation; Alternative splicing; AMPA; Desensitization; Flip and flop; Glutamate receptors

Indexed keywords

4 [2 (PHENYLSULFONYLAMINO)ETHYLTHIO] 2,6 DIFLUOROPHENOXYACETAMIDE; AMPA RECEPTOR; ANIRACETAM; CYCLOTHIAZIDE; GLUTAMATE RECEPTOR; PYROGLUTAMIC ACID; UNCLASSIFIED DRUG;

ALTERNATIVE RNA SPLICING; ARTICLE; DESENSITIZATION; DOSE RESPONSE; KINETICS; MEMBRANE CURRENT; NEUROMODULATION; OOCYTE; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 0030755886     PISSN: 02706474     EISSN: None     Source Type: Journal    
DOI: 10.1523/jneurosci.17-15-05760.1997     Document Type: Article

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