Pregna-D′-pentarane structure influences progesterone receptor affinity for DNA

Steroids

Volumn 67, Issue 5, 2002, Pages 323-332

  Shchelkunova, T A ^a   Rubtsov, P M ^b   Levina, I S ^c   Kamerntsky, A V ^c   Smirnov, A N ^a  

^a MOSCOW STATE UNIVERSITY   (Russian Federation)

^b ENGELHARDT INSTITUTE OF MOLECULAR BIOLOGY   (Russian Federation)

^c N D ZELINSKY INSTITUTE OF ORGANIC CHEMISTRY   (Russian Federation)

Author keywords

17 cycloalkane derivatives; DNA receptor affinity constants; Electrophoretic mobility shift assay; Hormone response element; Progesterone 16 ; Progesterone receptor

Indexed keywords

16ALPHA,17ALPHA CYCLOHEX 2' ENOPROGESTERONE; 16ALPHA,17ALPHA CYCLOHEXANOPROGESTERONE; 16ALPHA,17ALPHA CYCLOPENTANOPROGESTERONE; 16ALPHA,17ALPHA CYCLOPROPANOPROGESTERONE; 6ALPHA METHYL 16ALPHA,17ALPHA CYCLOHEXANOPROGESTERONE; DNA; MIFEPRISTONE; PROGESTERONE DERIVATIVE; PROGESTERONE RECEPTOR; PROMEGESTONE; TYROSINE AMINOTRANSFERASE; UNCLASSIFIED DRUG; DRUG DERIVATIVE; PRIMER DNA; PROGESTERONE;

ANIMAL TISSUE; ARTICLE; ASSAY; CONTROLLED STUDY; CYTOSOL; DNA PROTEIN COMPLEX; DNA SEQUENCE; DRUG ACTIVITY; ELECTROPHORETIC MOBILITY; FEMALE; HORMONE RESPONSIVE ELEMENT; NONHUMAN; RADIOACTIVITY; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; TEMPERATURE DEPENDENCE; ANIMAL; BINDING SITE; CHEMICAL STRUCTURE; CHEMISTRY; DNA RESPONSIVE ELEMENT; GEL MOBILITY SHIFT ASSAY; GENETICS; KINETICS; METABOLISM; PROMOTER REGION; TRANSACTIVATION; UTERUS; WISTAR RAT;

ANIMALS; BINDING SITES; CYTOSOL; DNA; DNA PRIMERS; ELECTROPHORETIC MOBILITY SHIFT ASSAY; FEMALE; KINETICS; MOLECULAR STRUCTURE; PROGESTERONE; PROMOTER REGIONS (GENETICS); RATS; RATS, WISTAR; RECEPTORS, PROGESTERONE; RESPONSE ELEMENTS; TRANS-ACTIVATION (GENETICS); TYROSINE TRANSAMINASE; UTERUS;

EID: 0036008937     PISSN: 0039128X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0039-128X(01)00188-X     Document Type: Article

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