Recent developments in combinatorial organic synthesis

Drug Discovery Today

Volumn 7, Issue 1, 2002, Pages 47-55

  Ganesan, A ^a  

^a UNIVERSITY OF SOUTHAMPTON   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

CARBAMIC ACID DERIVATIVE; GALANTAMINE; GUANIDINE DERIVATIVE; INDINAVIR; MACROLIDE; MEVINOLIN; NIFEDIPINE; OXAZOLIDINONE DERIVATIVE; PIPERIDINE DERIVATIVE; PYRROLE DERIVATIVE; SILDENAFIL; TACROLIMUS; VESAMICOL; VITAMIN D DERIVATIVE; ALIPHATIC HYDROCARBON; BIOLOGICAL FACTOR; HETEROCYCLIC COMPOUND; ALDEHYDE; CALCIUM CHANNEL BLOCKING AGENT; FK 506 BINDING PROTEIN; HYDROXYMETHYLGLUTARYL COENZYME A REDUCTASE INHIBITOR; IMMUNOSUPPRESSIVE AGENT; ION CHANNEL; NIFEDIPINE DERIVATIVE; PHOSPHODIESTERASE INHIBITOR; PROTEINASE INHIBITOR; RESIN; SCOPOLAMINE; SESQUITERPENE DERIVATIVE; TROPANONE; UNCLASSIFIED DRUG; VITAMIN D;

ALKYLATION; COMBINATORIAL CHEMISTRY; CYCLIZATION; DRUG ACTIVITY; DRUG SYNTHESIS; HYDROLYSIS; METHODOLOGY; PHARMACOPHORE; REVIEW; SOLID; CHEMISTRY; SYNTHESIS; CYCLOADDITION; DIELS ALDER REACTION; HORNER WADSWORTH EMMONS REACTION; MITSUNOBU REACTION;

BIOLOGICAL FACTORS; COMBINATORIAL CHEMISTRY TECHNIQUES; HETEROCYCLIC COMPOUNDS; HYDROCARBONS, ACYCLIC;

EID: 0036007206     PISSN: 13596446     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1359-6446(01)02087-6     Document Type: Review

References (24)

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3. Sequential nucleophilic substitution: A powerful strategy for the solid-phase production of diverse compound libraries
4. A combinatorial approach to polyketide-type libraries by iterative asymmetric aldol reactions performed on solid support
5. Polymer-aided stereodivergent synthesis (PASS): A new concept for the discrete preparation of optical antipodes
6. Solid-phase synthesis of 1,2,3,4-tetrahydro-2-pyridones via aza-annulation of enamines
7. Simple and efficient synthesis of 3,4-dihydro-2-pyridones via novel solid-supported aza-annulation
8. Combinatorial synthesis of libraries of indole derivatives
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13. Towards diversity-oriented, stereoselective syntheses of biaryl- or bis(aryl)metal-containing medium rings
14. Solid-phase Zincke route to pyridinium, tetrahydropyridine, and piperidine derivatives: Vesamicol analogs
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16. Parallel modification of tropane alkaloids
17. Synthesis and biological evaluation of a focused mixture library of analogues of the antimitotic marine natural product curacin A
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