Simple and efficient synthesis of 3,4-dihydro-2-pyridones via novel solid-supported aza-annulation

Journal of Organic Chemistry

Volumn 65, Issue 26, 2000, Pages 9103-9113

  Wagman, A S ^a   Wang, L ^a,b   Nuss, J M ^a,c  

^a NOVARTIS PHARMA AG   (Switzerland)

^b UNIVERSITY OF CALIFORNIA   (United States)

^c EXELIXIS INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETIC ACID; ACETOPHENONE; AMIDE; CHALCONE DERIVATIVE; METHYL 1 (2 FURYLMETHYL) 2 OXO 4 PHENYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYL 1 [2 [(6 CHLORO 2 FLUOROPHENYL)METHYLTHIO]ETHYL] 2 OXO 4 PHENYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYL 2 OXO 4 PHENYL 1 (2 PHENYLETHYL) 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYL 2 OXO 4 PHENYL 1 BENZYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYL 2 OXO 4 PHENYL 1 PROP 2 ENYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYL 2 OXO 4 PHENYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; METHYLMALONIC ACID; PROP 2 ENYL 2 OXO 4 PHENYL 1 BENZYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; PROP 2 ENYL 2 OXO 4 PHENYL 6 (4 SULFAMOYLPHENYL) 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; PROP 2 ENYL 4 (2,6 DICHLOROPHENYL) 6 (4 SULFAMOYLPHENYL) 2 OXO 1 BENZYL 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; PROP 2 ENYL 4 (3 NITROPHENYL) 6 (4 SULFAMOYLPHENYL) 2 OXO 1 BENZYL 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; PROP 2 ENYL 4 (4 CYANOPHENYL) 6 (4 SULFAMOYLPHENYL) 2 OXO 1 BENYZL 1,3,4 TRIHYDROPYRIDINE 3 CARBOXYLATE; PYRIDONE DERIVATIVE; RESIN; SULFONAMIDE; UNCLASSIFIED DRUG;

ARTICLE; CATALYST; CHEMICAL REACTION; CYCLIZATION; DRUG SYNTHESIS;

EID: 0034731531     PISSN: 00223263     EISSN: None     Source Type: Journal    
DOI: 10.1021/jo005609x     Document Type: Article

References (60)